De Jonghe S - Search Results

1

Design, synthesis, and molecular modeling studies of novel 2-quinolone-1,2,3-triazole-α-aminophosphonates hybrids as dual antiviral and antibacterial agents.

Gadali KE, Rafya M, El Mansouri AE, Maatallah M, Vanderlee A, Mehdi A, Neyts J, Jochmans D, De Jonghe S, Benkhalti F, Sanghvi YS, Taourirte M, Lazrek HB. Gadali KE, et al. Among authors: de jonghe s. Eur J Med Chem. 2024 Mar 15;268:116235. doi: 10.1016/j.ejmech.2024.116235. Epub 2024 Feb 16. Eur J Med Chem. 2024. PMID: 38377828 Review.

2

Discovery of 7-N-piperazinylthiazolo[5,4-d]pyrimidine analogues as a novel class of immunosuppressive agents with in vivo biological activity.

Jang MY, Lin Y, De Jonghe S, Gao LJ, Vanderhoydonck B, Froeyen M, Rozenski J, Herman J, Louat T, Van Belle K, Waer M, Herdewijn P. Jang MY, et al. Among authors: de jonghe s. J Med Chem. 2011 Jan 27;54(2):655-68. doi: 10.1021/jm101254z. Epub 2010 Dec 20. J Med Chem. 2011. PMID: 21171614

3

Discovery of dual death-associated protein related apoptosis inducing protein kinase 1 and 2 inhibitors by a scaffold hopping approach.

Gao LJ, Kovackova S, Sála M, Ramadori AT, De Jonghe S, Herdewijn P. Gao LJ, et al. Among authors: de jonghe s. J Med Chem. 2014 Sep 25;57(18):7624-43. doi: 10.1021/jm5007929. Epub 2014 Sep 11. J Med Chem. 2014. PMID: 25178155

4

Emimycin and its nucleoside derivatives: Synthesis and antiviral activity.

Plebanek E, Lescrinier E, Andrei G, Snoeck R, Herdewijn P, De Jonghe S. Plebanek E, et al. Among authors: de jonghe s. Eur J Med Chem. 2018 Jan 20;144:93-103. doi: 10.1016/j.ejmech.2017.12.018. Epub 2017 Dec 7. Eur J Med Chem. 2018. PMID: 29268134

5

Synthesis and antiviral evaluation of cyclopentyl nucleoside phosphonates.

Wang M, Srivastava P, Liu C, Snoeck R, Andrei G, De Jonghe S, Herdewijn P. Wang M, et al. Among authors: de jonghe s. Eur J Med Chem. 2018 Apr 25;150:616-625. doi: 10.1016/j.ejmech.2018.03.008. Epub 2018 Mar 10. Eur J Med Chem. 2018. PMID: 29550734

6

Cyclin G-associated kinase (GAK) affinity and antiviral activity studies of a series of 3-C-substituted isothiazolo[4,3-b]pyridines.

Wouters R, Pu SY, Froeyen M, Lescrinier E, Einav S, Herdewijn P, De Jonghe S. Wouters R, et al. Among authors: de jonghe s. Eur J Med Chem. 2019 Feb 1;163:256-265. doi: 10.1016/j.ejmech.2018.11.065. Epub 2018 Nov 28. Eur J Med Chem. 2019. PMID: 30529544

7

Design, synthesis and biological evaluation of pyrazolo[3,4-d]pyrimidine-based protein kinase D inhibitors.

Gilles P, Kashyap RS, Freitas MJ, Ceusters S, Van Asch K, Janssens A, De Jonghe S, Persoons L, Cobbaut M, Daelemans D, Van Lint J, Voet ARD, De Borggraeve WM. Gilles P, et al. Among authors: de jonghe s, de borggraeve wm. Eur J Med Chem. 2020 Nov 1;205:112638. doi: 10.1016/j.ejmech.2020.112638. Epub 2020 Jul 29. Eur J Med Chem. 2020. PMID: 32835918

8

Discovery of 3-phenyl- and 3-N-piperidinyl-isothiazolo[4,3-b]pyridines as highly potent inhibitors of cyclin G-associated kinase.

Martinez-Gualda B, Saul S, Froeyen M, Schols D, Herdewijn P, Einav S, De Jonghe S. Martinez-Gualda B, et al. Among authors: de jonghe s. Eur J Med Chem. 2021 Mar 5;213:113158. doi: 10.1016/j.ejmech.2021.113158. Epub 2021 Jan 12. Eur J Med Chem. 2021. PMID: 33497888

9

Kobophenol A Inhibits Binding of Host ACE2 Receptor with Spike RBD Domain of SARS-CoV-2, a Lead Compound for Blocking COVID-19.

Gangadevi S, Badavath VN, Thakur A, Yin N, De Jonghe S, Acevedo O, Jochmans D, Leyssen P, Wang K, Neyts J, Yujie T, Blum G. Gangadevi S, et al. Among authors: de jonghe s. J Phys Chem Lett. 2021 Feb 25;12(7):1793-1802. doi: 10.1021/acs.jpclett.0c03119. Epub 2021 Feb 12. J Phys Chem Lett. 2021. PMID: 33577324

10

In vitro activity of itraconazole against SARS-CoV-2.

Van Damme E, De Meyer S, Bojkova D, Ciesek S, Cinatl J, De Jonghe S, Jochmans D, Leyssen P, Buyck C, Neyts J, Van Loock M. Van Damme E, et al. Among authors: de jonghe s, de meyer s. J Med Virol. 2021 Jul;93(7):4454-4460. doi: 10.1002/jmv.26917. J Med Virol. 2021. PMID: 33666253 Free PMC article.

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