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Discovery and Development of Quinazolinones and Quinazolinediones for Ameliorating Nonalcoholic Fatty Liver Disease (NAFLD) by Modulating COP1-ATGL Axis.
J Med Chem. 2023 Dec 28;66(24):16728-16761. doi: 10.1021/acs.jmedchem.3c01431. Epub 2023 Dec 15.
J Med Chem. 2023.
PMID: 38100045
Mitigating hERG Liability of Toll-Like Receptor 9 and 7 Antagonists through Structure-Based Design.
Das N, Bhattacharya D, Bandopadhyay P, Dastidar UG, Paul B, Rahaman O, Hoque I, Patra B, Ganguly D, Talukdar A.
Das N, et al. Among authors: dastidar ug.
ChemMedChem. 2023 Jun 15;18(12):e202300069. doi: 10.1002/cmdc.202300069. Epub 2023 Apr 18.
ChemMedChem. 2023.
PMID: 36999630
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Development, Optimization, and In Vivo Validation of New Imidazopyridine Chemotypes as Dual TLR7/TLR9 Antagonists through Activity-Directed Sequential Incorporation of Relevant Structural Subunits.
Das N, Bandopadhyay P, Roy S, Sinha BP, Dastidar UG, Rahaman O, Pal S, Ganguly D, Talukdar A.
Das N, et al. Among authors: dastidar ug.
J Med Chem. 2022 Sep 8;65(17):11607-11632. doi: 10.1021/acs.jmedchem.2c00386. Epub 2022 Aug 12.
J Med Chem. 2022.
PMID: 35959635
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