D'Ascenzio M - Search Results

1

Opening New Scenarios for Human MAO Inhibitors.

De Monte C, D'Ascenzio M, Guglielmi P, Mancini V, Carradori S. De Monte C, et al. Among authors: d ascenzio m. Cent Nerv Syst Agents Med Chem. 2016;16(2):98-104. doi: 10.2174/1871524915666150831141705. Cent Nerv Syst Agents Med Chem. 2016. PMID: 26320583 Review.

2

Synthesis and selective human monoamine oxidase B inhibition of heterocyclic hybrids based on hydrazine and thiazole scaffolds.

Carradori S, D'Ascenzio M, De Monte C, Secci D, Yáñez M. Carradori S, et al. Arch Pharm (Weinheim). 2013 Jan;346(1):17-22. doi: 10.1002/ardp.201200318. Epub 2012 Oct 15. Arch Pharm (Weinheim). 2013. PMID: 23065686

3

Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors.

D'Ascenzio M, Carradori S, Secci D, Mannina L, Sobolev AP, De Monte C, Cirilli R, Yáñez M, Alcaro S, Ortuso F. D'Ascenzio M, et al. Bioorg Med Chem. 2014 May 15;22(10):2887-95. doi: 10.1016/j.bmc.2014.03.042. Epub 2014 Apr 5. Bioorg Med Chem. 2014. PMID: 24746464

4

(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.

D'Ascenzio M, Chimenti P, Gidaro MC, De Monte C, De Vita D, Granese A, Scipione L, Di Santo R, Costa G, Alcaro S, Yáñez M, Carradori S. D'Ascenzio M, et al. J Enzyme Inhib Med Chem. 2015 Dec;30(6):908-19. doi: 10.3109/14756366.2014.987138. Epub 2015 Sep 25. J Enzyme Inhib Med Chem. 2015. PMID: 25807300

5

New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: biological evaluation and molecular modelling studies.

Carradori S, Mollica A, Ceruso M, D'Ascenzio M, De Monte C, Chimenti P, Sabia R, Akdemir A, Supuran CT. Carradori S, et al. Among authors: d ascenzio m. Bioorg Med Chem. 2015 Jul 1;23(13):2975-81. doi: 10.1016/j.bmc.2015.05.013. Epub 2015 May 14. Bioorg Med Chem. 2015. PMID: 26007302

6

Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential.

Carradori S, Secci D, Bolasco A, Chimenti P, D'Ascenzio M. Carradori S, et al. Expert Opin Ther Pat. 2012 Jul;22(7):759-801. doi: 10.1517/13543776.2012.698613. Epub 2012 Jun 18. Expert Opin Ther Pat. 2012. PMID: 22702491 Review.

7

Recent advances in the development of selective human MAO-B inhibitors: (hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines.

Secci D, Bolasco A, Carradori S, D'Ascenzio M, Nescatelli R, Yáñez M. Secci D, et al. Eur J Med Chem. 2012 Dec;58:405-17. doi: 10.1016/j.ejmech.2012.10.032. Epub 2012 Oct 26. Eur J Med Chem. 2012. PMID: 23153812

8

Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors.

Secci D, Carradori S, Bolasco A, Bizzarri B, D'Ascenzio M, Maccioni E. Secci D, et al. Curr Top Med Chem. 2012;12(20):2240-57. doi: 10.2174/156802612805220057. Curr Top Med Chem. 2012. PMID: 23276158 Review.

9

Exploring 4-substituted-2-thiazolylhydrazones from 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors.

Chimenti P, Petzer A, Carradori S, D'Ascenzio M, Silvestri R, Alcaro S, Ortuso F, Petzer JP, Secci D. Chimenti P, et al. Eur J Med Chem. 2013 Aug;66:221-7. doi: 10.1016/j.ejmech.2013.05.032. Epub 2013 Jun 3. Eur J Med Chem. 2013. PMID: 23807114

10

Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII--a new scaffold for designing isoform-selective inhibitors.

Carradori S, De Monte C, D'Ascenzio M, Secci D, Celik G, Ceruso M, Vullo D, Scozzafava A, Supuran CT. Carradori S, et al. Bioorg Med Chem Lett. 2013 Dec 15;23(24):6759-63. doi: 10.1016/j.bmcl.2013.10.026. Epub 2013 Oct 26. Bioorg Med Chem Lett. 2013. PMID: 24189056

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