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Blockage of A2A and A3 adenosine receptors decreases the desensitization of human GABA(A) receptors microtransplanted to Xenopus oocytes.
Roseti C, Palma E, Martinello K, Fucile S, Morace R, Esposito V, Cantore G, Arcella A, Giangaspero F, Aronica E, Mascia A, Di Gennaro G, Quarato PP, Manfredi M, Cristalli G, Lambertucci C, Marucci G, Volpini R, Limatola C, Eusebi F. Roseti C, et al. Among authors: cristalli g. Proc Natl Acad Sci U S A. 2009 Sep 15;106(37):15927-31. doi: 10.1073/pnas.0907324106. Epub 2009 Aug 31. Proc Natl Acad Sci U S A. 2009. PMID: 19721003 Free PMC article.
P2 receptor antagonists prevent synaptic failure and extracellular signal-regulated kinase 1/2 activation induced by oxygen and glucose deprivation in rat CA1 hippocampus in vitro.
Traini C, Pedata F, Cipriani S, Mello T, Galli A, Giovannini MG, Cerbai F, Volpini R, Cristalli G, Pugliese AM. Traini C, et al. Among authors: cristalli g. Eur J Neurosci. 2011 Jun;33(12):2203-15. doi: 10.1111/j.1460-9568.2011.07667.x. Epub 2011 Apr 1. Eur J Neurosci. 2011. PMID: 21453436
Pyrazolo[1,5-c]quinazoline derivatives and their simplified analogues as adenosine receptor antagonists: synthesis, structure-affinity relationships and molecular modeling studies.
Catarzi D, Colotta V, Varano F, Poli D, Squarcialupi L, Filacchioni G, Varani K, Vincenzi F, Borea PA, Dal Ben D, Lambertucci C, Cristalli G. Catarzi D, et al. Among authors: cristalli g. Bioorg Med Chem. 2013 Jan 1;21(1):283-94. doi: 10.1016/j.bmc.2012.10.031. Epub 2012 Oct 29. Bioorg Med Chem. 2013. PMID: 23171656
Synthesis, structure-affinity relationships, and molecular modeling studies of novel pyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists.
Lenzi O, Colotta V, Catarzi D, Varano F, Squarcialupi L, Filacchioni G, Varani K, Vincenzi F, Borea PA, Dal Ben D, Lambertucci C, Cristalli G. Lenzi O, et al. Among authors: cristalli g. Bioorg Med Chem. 2011 Jun 15;19(12):3757-68. doi: 10.1016/j.bmc.2011.05.001. Epub 2011 May 6. Bioorg Med Chem. 2011. PMID: 21616671
Adenosine derivatives as agonists of adenosine receptors.
Grifantini M, Cristalli G, Franchetti P, Vittori S. Grifantini M, et al. Among authors: cristalli g. Farmaco. 1991 Jan;46(1 Suppl):161-9. Farmaco. 1991. PMID: 1854403 Review. No abstract available.
212 results