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New BACE1 Chimeric Peptide Inhibitors Selectively Prevent AβPP-β Cleavage Decreasing Amyloid-β Production and Accumulation in Alzheimer's Disease Models.
J Alzheimers Dis. 2020;76(4):1317-1337. doi: 10.3233/JAD-200381.
J Alzheimers Dis. 2020.
PMID: 32597812
Highlights in BACE1 Inhibitors for Alzheimer's Disease Treatment.
Coimbra JRM, Marques DFF, Baptista SJ, Pereira CMF, Moreira PI, Dinis TCP, Santos AE, Salvador JAR.
Coimbra JRM, et al.
Front Chem. 2018 May 24;6:178. doi: 10.3389/fchem.2018.00178. eCollection 2018.
Front Chem. 2018.
PMID: 29881722
Free PMC article.
Review.
Item in Clipboard
An overview of glutaminyl cyclase inhibitors for Alzheimer's disease.
Coimbra JR, Sobral PJ, Santos AE, Moreira PI, Salvador JA.
Coimbra JR, et al.
Future Med Chem. 2019 Dec;11(24):3179-3194. doi: 10.4155/fmc-2019-0163.
Future Med Chem. 2019.
PMID: 31838899
Review.
Item in Clipboard
Combining Virtual Screening Protocol and In Vitro Evaluation towards the Discovery of BACE1 Inhibitors.
Coimbra JRM, Baptista SJ, Dinis TCP, Silva MMC, Moreira PI, Santos AE, Salvador JAR.
Coimbra JRM, et al.
Biomolecules. 2020 Apr 1;10(4):535. doi: 10.3390/biom10040535.
Biomolecules. 2020.
PMID: 32244832
Free PMC article.
Item in Clipboard
A patent review of glutaminyl cyclase inhibitors (2004-present).
Coimbra JRM, Salvador JAR.
Coimbra JRM, et al.
Expert Opin Ther Pat. 2021 Sep;31(9):809-836. doi: 10.1080/13543776.2021.1917549. Epub 2021 Jul 5.
Expert Opin Ther Pat. 2021.
PMID: 33896339
Review.
Item in Clipboard
Therapeutic potential of glutaminyl cyclases: Current status and emerging trends.
Coimbra JRM, Moreira PI, Santos AE, Salvador JAR.
Coimbra JRM, et al.
Drug Discov Today. 2023 Oct;28(10):103644. doi: 10.1016/j.drudis.2023.103644. Epub 2023 May 26.
Drug Discov Today. 2023.
PMID: 37244566
Free article.
Review.
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