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Antitumor activity of novel POLA1-HDAC11 dual inhibitors.
Dallavalle S, Musso L, Cincinelli R, Darwiche N, Gervasoni S, Vistoli G, Guglielmi MB, La Porta I, Pizzulo M, Modica E, Prosperi F, Signorino G, Colelli F, Cardile F, Fucci A, D'Andrea EL, Riccio A, Pisano C. Dallavalle S, et al. Among authors: cincinelli r. Eur J Med Chem. 2022 Jan 15;228:113971. doi: 10.1016/j.ejmech.2021.113971. Epub 2021 Nov 3. Eur J Med Chem. 2022. PMID: 34772529
7-Azaindole-1-carboxamides as a new class of PARP-1 inhibitors.
Cincinelli R, Musso L, Merlini L, Giannini G, Vesci L, Milazzo FM, Carenini N, Perego P, Penco S, Artali R, Zunino F, Pisano C, Dallavalle S. Cincinelli R, et al. Bioorg Med Chem. 2014 Feb 1;22(3):1089-103. doi: 10.1016/j.bmc.2013.12.031. Epub 2013 Dec 22. Bioorg Med Chem. 2014. PMID: 24398383 Free article.
Hybrid topoisomerase I and HDAC inhibitors as dual action anticancer agents.
Cincinelli R, Musso L, Artali R, Guglielmi MB, La Porta I, Melito C, Colelli F, Cardile F, Signorino G, Fucci A, Frusciante M, Pisano C, Dallavalle S. Cincinelli R, et al. PLoS One. 2018 Oct 9;13(10):e0205018. doi: 10.1371/journal.pone.0205018. eCollection 2018. PLoS One. 2018. PMID: 30300374 Free PMC article.
Novel adamantyl retinoid-related molecules with POLA1 inhibitory activity.
Cincinelli R, Musso L, Guglielmi MB, La Porta I, Fucci A, Luca D'Andrea E, Cardile F, Colelli F, Signorino G, Darwiche N, Gervasoni S, Vistoli G, Pisano C, Dallavalle S. Cincinelli R, et al. Bioorg Chem. 2020 Nov;104:104253. doi: 10.1016/j.bioorg.2020.104253. Epub 2020 Sep 2. Bioorg Chem. 2020. PMID: 32920362
26 results