Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
7 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Tacrine - Benzothiazoles: Novel class of potential multitarget anti-Alzheimeŕs drugs dealing with cholinergic, amyloid and mitochondrial systems.
Bioorg Chem. 2021 Feb;107:104596. doi: 10.1016/j.bioorg.2020.104596. Epub 2020 Dec 28.
Bioorg Chem. 2021.
PMID: 33421953
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease.
Chalupova K, Korabecny J, Bartolini M, Monti B, Lamba D, Caliandro R, Pesaresi A, Brazzolotto X, Gastellier AJ, Nachon F, Pejchal J, Jarosova M, Hepnarova V, Jun D, Hrabinova M, Dolezal R, Zdarova Karasova J, Mzik M, Kristofikova Z, Misik J, Muckova L, Jost P, Soukup O, Benkova M, Setnicka V, Habartova L, Chvojkova M, Kleteckova L, Vales K, Mezeiova E, Uliassi E, Valis M, Nepovimova E, Bolognesi ML, Kuca K.
Chalupova K, et al.
Eur J Med Chem. 2019 Apr 15;168:491-514. doi: 10.1016/j.ejmech.2019.02.021. Epub 2019 Feb 27.
Eur J Med Chem. 2019.
PMID: 30851693
Item in Clipboard
Huprine Y - Tryptophan heterodimers with potential implication to Alzheimer's disease treatment.
Mezeiova E, Hrabinova M, Hepnarova V, Jun D, Janockova J, Muckova L, Prchal L, Kristofikova Z, Kucera T, Gorecki L, Chalupova K, Kunes J, Hroudova J, Soukup O, Korabecny J.
Mezeiova E, et al. Among authors: chalupova k.
Bioorg Med Chem Lett. 2021 Jul 1;43:128100. doi: 10.1016/j.bmcl.2021.128100. Epub 2021 May 10.
Bioorg Med Chem Lett. 2021.
PMID: 33984470
Item in Clipboard
Donepezil Derivatives Targeting Amyloid-β Cascade in Alzheimer's Disease.
Mezeiova E, Chalupova K, Nepovimova E, Gorecki L, Prchal L, Malinak D, Kuca K, Soukup O, Korabecny J.
Mezeiova E, et al. Among authors: chalupova k.
Curr Alzheimer Res. 2019;16(9):772-800. doi: 10.2174/1567205016666190228122956.
Curr Alzheimer Res. 2019.
PMID: 30819078
Review.
Item in Clipboard
UHPLC-HRMS study of anti-Alzheimer's drug candidates: metabolism of 7-MEOTA-tryptophan hybrids hampers their passage into brain.
Mžik M, Žďárová-Karasová J, Chalupová K, Korábečný J, Palička V, Šesták V.
Mžik M, et al. Among authors: chalupova k.
J Pharm Biomed Anal. 2019 Sep 10;174:134-144. doi: 10.1016/j.jpba.2019.05.051. Epub 2019 May 24.
J Pharm Biomed Anal. 2019.
PMID: 31167157
Item in Clipboard
Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition.
Oleksak P, Psotka M, Vancurova M, Sapega O, Bieblova J, Reinis M, Rysanek D, Mikyskova R, Chalupova K, Malinak D, Svobodova J, Andrys R, Rehulkova H, Skopek V, Ngoc Lam P, Bartek J, Hodny Z, Musilek K.
Oleksak P, et al. Among authors: chalupova k.
J Enzyme Inhib Med Chem. 2021 Dec;36(1):410-424. doi: 10.1080/14756366.2020.1871336.
J Enzyme Inhib Med Chem. 2021.
PMID: 33440995
Free PMC article.
Item in Clipboard
Nanomolar Benzothiazole-Based Inhibitors of 17β-HSD10 with Cellular Bioactivity.
Hanzlova M, Miskerikova MS, Rotterova A, Chalupova K, Jurkova K, Hamsikova M, Andrys R, Haleckova A, Svobodova J, Schmidt M, Benek O, Musilek K.
Hanzlova M, et al. Among authors: chalupova k.
ACS Med Chem Lett. 2023 Nov 10;14(12):1724-1732. doi: 10.1021/acsmedchemlett.3c00355. eCollection 2023 Dec 14.
ACS Med Chem Lett. 2023.
PMID: 38116418
Item in Clipboard
Cite
Cite