Synthesis of a CGRP Receptor Antagonist via an Asymmetric Synthesis of 3-Fluoro-4-aminopiperidine.
Molinaro C, Phillips EM, Xiang B, Milczek E, Shevlin M, Balsells J, Ceglia S, Chen J, Chen L, Chen Q, Fei Z, Hoerrner S, Qi J, de Lera Ruiz M, Tan L, Wan B, Yin J.
Molinaro C, et al. Among authors: ceglia s.
J Org Chem. 2019 Jun 21;84(12):8006-8018. doi: 10.1021/acs.joc.9b00569. Epub 2019 Jun 5.
J Org Chem. 2019.
PMID: 31124362