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Antivascular and antitumor properties of the tubulin-binding chalcone TUB091.
Oncotarget. 2017 Feb 28;8(9):14325-14342. doi: 10.18632/oncotarget.9527.
Oncotarget. 2017.
PMID: 27224920
Free PMC article.
Novel colchicine-site binders with a cyclohexanedione scaffold identified through a ligand-based virtual screening approach.
Canela MD, Pérez-Pérez MJ, Noppen S, Sáez-Calvo G, Díaz JF, Camarasa MJ, Liekens S, Priego EM.
Canela MD, et al.
J Med Chem. 2014 May 22;57(10):3924-38. doi: 10.1021/jm401939g. Epub 2014 May 9.
J Med Chem. 2014.
PMID: 24773591
Free article.
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Blocking Blood Flow to Solid Tumors by Destabilizing Tubulin: An Approach to Targeting Tumor Growth.
Pérez-Pérez MJ, Priego EM, Bueno O, Martins MS, Canela MD, Liekens S.
Pérez-Pérez MJ, et al. Among authors: canela md.
J Med Chem. 2016 Oct 13;59(19):8685-8711. doi: 10.1021/acs.jmedchem.6b00463. Epub 2016 Jun 27.
J Med Chem. 2016.
PMID: 27348355
Free article.
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Identification of [1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-ones as novel inhibitors of Chikungunya virus replication.
Gigante A, Canela MD, Delang L, Priego EM, Camarasa MJ, Querat G, Neyts J, Leyssen P, Pérez-Pérez MJ.
Gigante A, et al. Among authors: canela md.
J Med Chem. 2014 May 22;57(10):4000-8. doi: 10.1021/jm401844c. Epub 2014 May 6.
J Med Chem. 2014.
PMID: 24800626
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Synthesis and antiproliferative activity of 6-phenylaminopurines.
Canela MD, Liekens S, Camarasa MJ, Priego EM, Pérez-Pérez MJ.
Canela MD, et al.
Eur J Med Chem. 2014 Nov 24;87:421-8. doi: 10.1016/j.ejmech.2014.09.093. Epub 2014 Sep 30.
Eur J Med Chem. 2014.
PMID: 25282265
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Efficient synthesis and anti-enteroviral activity of 9-arylpurines.
Aguado L, Canela MD, Thibaut HJ, Priego EM, Camarasa MJ, Leyssen P, Neyts J, Pérez-Pérez MJ.
Aguado L, et al. Among authors: canela md.
Eur J Med Chem. 2012 Mar;49:279-88. doi: 10.1016/j.ejmech.2012.01.022. Epub 2012 Jan 17.
Eur J Med Chem. 2012.
PMID: 22305341
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Binding of glutathione to enterovirus capsids is essential for virion morphogenesis.
Thibaut HJ, van der Linden L, Jiang P, Thys B, Canela MD, Aguado L, Rombaut B, Wimmer E, Paul A, Pérez-Pérez MJ, van Kuppeveld FJ, Neyts J.
Thibaut HJ, et al. Among authors: canela md.
PLoS Pathog. 2014 Apr 10;10(4):e1004039. doi: 10.1371/journal.ppat.1004039. eCollection 2014 Apr.
PLoS Pathog. 2014.
PMID: 24722756
Free PMC article.
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