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Identification of inhibitors targeting the energy-coupling factor (ECF) transporters.
Commun Biol. 2023 Nov 20;6(1):1182. doi: 10.1038/s42003-023-05555-x.
Commun Biol. 2023.
PMID: 37985798
Free PMC article.
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay.
Bousis S, Winkler S, Haupenthal J, Fulco F, Diamanti E, Hirsch AKH.
Bousis S, et al.
Int J Mol Sci. 2022 Feb 27;23(5):2637. doi: 10.3390/ijms23052637.
Int J Mol Sci. 2022.
PMID: 35269783
Free PMC article.
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Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters.
Kiefer AF, Bousis S, Hamed MM, Diamanti E, Haupenthal J, Hirsch AKH.
Kiefer AF, et al. Among authors: bousis s.
J Med Chem. 2022 Jul 14;65(13):8869-8880. doi: 10.1021/acs.jmedchem.1c02114. Epub 2022 Jun 16.
J Med Chem. 2022.
PMID: 35709475
Free PMC article.
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Author Correction: Identification of inhibitors targeting the energy-coupling factor (ECF) transporters.
Diamanti E, Souza PCT, Setyawati I, Bousis S, Monjas L, Swier LJYM, Shams A, Tsarenko A, Stanek WK, Jäger M, Marrink SJ, Slotboom DJ, Hirsch AKH.
Diamanti E, et al. Among authors: bousis s.
Commun Biol. 2024 Jan 9;7(1):70. doi: 10.1038/s42003-024-05770-0.
Commun Biol. 2024.
PMID: 38195913
Free PMC article.
No abstract available.
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Synthesis and biological studies of c(RGDyK) conjugates of cucurbitacins.
Chatzisideri T, Dalezis P, Leonidis G, Bousis S, Trafalis D, Bianchini F, Sarli V.
Chatzisideri T, et al. Among authors: bousis s.
Future Med Chem. 2021 May;13(10):877-895. doi: 10.4155/fmc-2020-0309. Epub 2021 Apr 16.
Future Med Chem. 2021.
PMID: 33858195
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