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Novel S1P1 receptor agonists - Part 5: From amino-to alkoxy-pyridines.
Eur J Med Chem. 2016 Jun 10;115:326-41. doi: 10.1016/j.ejmech.2016.03.020. Epub 2016 Mar 12.
Eur J Med Chem. 2016.
PMID: 27027817
Novel S1P1 receptor agonists--part 1: From pyrazoles to thiophenes.
Bolli MH, Müller C, Mathys B, Abele S, Birker M, Bravo R, Bur D, Hess P, Kohl C, Lehmann D, Nayler O, Rey M, Meyer S, Scherz M, Schmidt G, Steiner B, Treiber A, Velker J, Weller T.
Bolli MH, et al. Among authors: birker m.
J Med Chem. 2013 Dec 12;56(23):9737-55. doi: 10.1021/jm4014373. Epub 2013 Nov 22.
J Med Chem. 2013.
PMID: 24266709
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Novel S1P(1) receptor agonists--part 2: from bicyclo[3.1.0]hexane-fused thiophenes to isobutyl substituted thiophenes.
Bolli MH, Velker J, Müller C, Mathys B, Birker M, Bravo R, Bur D, de Kanter R, Hess P, Kohl C, Lehmann D, Meyer S, Nayler O, Rey M, Scherz M, Steiner B.
Bolli MH, et al. Among authors: birker m.
J Med Chem. 2014 Jan 9;57(1):78-97. doi: 10.1021/jm401456d. Epub 2013 Dec 17.
J Med Chem. 2014.
PMID: 24345087
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Novel S1P(1) receptor agonists--part 3: from thiophenes to pyridines.
Bolli MH, Abele S, Birker M, Bravo R, Bur D, de Kanter R, Kohl C, Grimont J, Hess P, Lescop C, Mathys B, Müller C, Nayler O, Rey M, Scherz M, Schmidt G, Seifert J, Steiner B, Velker J, Weller T.
Bolli MH, et al. Among authors: birker m.
J Med Chem. 2014 Jan 9;57(1):110-30. doi: 10.1021/jm4014696. Epub 2013 Dec 24.
J Med Chem. 2014.
PMID: 24367923
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Novel S1P1 receptor agonists - Part 4: Alkylaminomethyl substituted aryl head groups.
Lescop C, Müller C, Mathys B, Birker M, de Kanter R, Kohl C, Hess P, Nayler O, Rey M, Sieber P, Steiner B, Weller T, Bolli MH.
Lescop C, et al. Among authors: birker m.
Eur J Med Chem. 2016 Jun 30;116:222-238. doi: 10.1016/j.ejmech.2016.03.048. Epub 2016 Mar 23.
Eur J Med Chem. 2016.
PMID: 27061986
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Discovery of the Novel, Orally Active, and Selective LPA1 Receptor Antagonist ACT-1016-0707 as a Preclinical Candidate for the Treatment of Fibrotic Diseases.
Lescop C, Birker M, Brotschi C, Bürki C, Morrison K, Froidevaux S, Delahaye S, Nayler O, Bolli MH.
Lescop C, et al. Among authors: birker m.
J Med Chem. 2024 Feb 22;67(4):2397-2424. doi: 10.1021/acs.jmedchem.3c01827. Epub 2024 Feb 13.
J Med Chem. 2024.
PMID: 38349250
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Discovery of a Novel Orally Active, Selective LPA Receptor Type 1 Antagonist, 4-(4-(2-Isopropylphenyl)-4-((2-methoxy-4-methylphenyl)carbamoyl)piperidin-1-yl)-4-oxobutanoic Acid, with a Distinct Molecular Scaffold.
Lescop C, Brotschi C, Williams JT, Sager CP, Birker M, Morrison K, Froidevaux S, Delahaye S, Nayler O, Bolli MH.
Lescop C, et al. Among authors: birker m.
J Med Chem. 2024 Feb 22;67(4):2379-2396. doi: 10.1021/acs.jmedchem.3c01826. Epub 2024 Feb 13.
J Med Chem. 2024.
PMID: 38349223
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The effect of ambient temperature, habitat quality and individual age on incubation behaviour and incubation feeding in a socially monogamous songbird.
Amininasab SM, Kingma SA, Birker M, Hildenbrandt H, Komdeur J.
Amininasab SM, et al. Among authors: birker m.
Behav Ecol Sociobiol. 2016;70:1591-1600. doi: 10.1007/s00265-016-2167-2. Epub 2016 Jul 5.
Behav Ecol Sociobiol. 2016.
PMID: 27546954
Free PMC article.
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