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Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors.
Bioorg Med Chem Lett. 2022 Jan 1;55:128449. doi: 10.1016/j.bmcl.2021.128449. Epub 2021 Nov 12.
Bioorg Med Chem Lett. 2022.
PMID: 34780899
Synthesis and biological evaluation of 3-substituted 2-oxindole derivatives as new glycogen synthase kinase 3β inhibitors.
Lozinskaya NA, Babkov DA, Zaryanova EV, Bezsonova EN, Efremov AM, Tsymlyakov MD, Anikina LV, Zakharyascheva OY, Borisov AV, Perfilova VN, Tyurenkov IN, Proskurnina MV, Spasov AA.
Lozinskaya NA, et al. Among authors: bezsonova en.
Bioorg Med Chem. 2019 May 1;27(9):1804-1817. doi: 10.1016/j.bmc.2019.03.028. Epub 2019 Mar 15.
Bioorg Med Chem. 2019.
PMID: 30902399
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Synthesis of New 2,3-Dihydroindole Derivatives and Evaluation of Their Melatonin Receptor Binding Affinity.
Volkova MS, Efremov AM, Bezsonova EN, Tsymliakov MD, Maksutova AI, Salykina MA, Sosonyuk SE, Shevtsova EF, Lozinskaya NA.
Volkova MS, et al. Among authors: bezsonova en.
Molecules. 2022 Nov 2;27(21):7462. doi: 10.3390/molecules27217462.
Molecules. 2022.
PMID: 36364290
Free PMC article.
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3-Arylidene-2-oxindoles as Potent NRH:Quinone Oxidoreductase 2 Inhibitors.
Lozinskaya NA, Bezsonova EN, Dubar M, Melekhina DD, Bazanov DR, Bunev AS, Grigor'eva OB, Klochkov VG, Sokolova EV, Babkov DA, Spasov AA, Sosonyuk SE.
Lozinskaya NA, et al. Among authors: bezsonova en.
Molecules. 2023 Jan 25;28(3):1174. doi: 10.3390/molecules28031174.
Molecules. 2023.
PMID: 36770840
Free PMC article.
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3-Arylidene-2-oxindoles as GSK3β inhibitors and anti-thrombotic agents.
Babkov D, Bezsonova E, Sirotenko V, Othman E, Klochkov V, Sosonyuk S, Lozinskaya N, Spasov A.
Babkov D, et al.
Bioorg Med Chem Lett. 2023 May 1;87:129283. doi: 10.1016/j.bmcl.2023.129283. Epub 2023 Apr 11.
Bioorg Med Chem Lett. 2023.
PMID: 37054760
Free PMC article.
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