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Novel Aminoquinoline Derivatives Significantly Reduce Parasite Load in Leishmania infantum Infected Mice.
Konstantinović J, Videnović M, Orsini S, Bogojević K, D'Alessandro S, Scaccabarozzi D, Terzić Jovanović N, Gradoni L, Basilico N, Šolaja BA. Konstantinović J, et al. Among authors: basilico n. ACS Med Chem Lett. 2018 May 4;9(7):629-634. doi: 10.1021/acsmedchemlett.8b00053. eCollection 2018 Jul 12. ACS Med Chem Lett. 2018. PMID: 30034591 Free PMC article.
Antimalarial activity of novel pyrrolizidinyl derivatives of 4-aminoquinoline.
Sparatore A, Basilico N, Casagrande M, Parapini S, Taramelli D, Brun R, Wittlin S, Sparatore F. Sparatore A, et al. Among authors: basilico n. Bioorg Med Chem Lett. 2008 Jul 1;18(13):3737-40. doi: 10.1016/j.bmcl.2008.05.042. Epub 2008 May 16. Bioorg Med Chem Lett. 2008. PMID: 18538567
A chemotype that inhibits three unrelated pathogenic targets: the botulinum neurotoxin serotype A light chain, P. falciparum malaria, and the Ebola filovirus.
Opsenica I, Burnett JC, Gussio R, Opsenica D, Todorović N, Lanteri CA, Sciotti RJ, Gettayacamin M, Basilico N, Taramelli D, Nuss JE, Wanner L, Panchal RG, Solaja BA, Bavari S. Opsenica I, et al. Among authors: basilico n. J Med Chem. 2011 Mar 10;54(5):1157-69. doi: 10.1021/jm100938u. Epub 2011 Jan 25. J Med Chem. 2011. PMID: 21265542 Free PMC article.
Hypoxia modulates the effect of dihydroartemisinin on endothelial cells.
D'Alessandro S, Basilico N, Corbett Y, Scaccabarozzi D, Omodeo-Salè F, Saresella M, Marventano I, Vaillant M, Olliaro P, Taramelli D. D'Alessandro S, et al. Among authors: basilico n. Biochem Pharmacol. 2011 Sep 1;82(5):476-84. doi: 10.1016/j.bcp.2011.06.002. Epub 2011 Jun 13. Biochem Pharmacol. 2011. PMID: 21684264
Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: further structure-activity relationships, in vivo studies, and preliminary toxicity profiling.
Gemma S, Camodeca C, Sanna Coccone S, Joshi BP, Bernetti M, Moretti V, Brogi S, Bonache de Marcos MC, Savini L, Taramelli D, Basilico N, Parapini S, Rottmann M, Brun R, Lamponi S, Caccia S, Guiso G, Summers RL, Martin RE, Saponara S, Gorelli B, Novellino E, Campiani G, Butini S. Gemma S, et al. Among authors: basilico n. J Med Chem. 2012 Aug 9;55(15):6948-67. doi: 10.1021/jm300802s. Epub 2012 Jul 27. J Med Chem. 2012. PMID: 22783984
Antiplasmodial activities of 4-aminoquinoline-statine compounds.
Vaiana N, Marzahn M, Parapini S, Liu P, Dell'Agli M, Pancotti A, Sangiovanni E, Basilico N, Bosisio E, Dunn BM, Taramelli D, Romeo S. Vaiana N, et al. Among authors: basilico n. Bioorg Med Chem Lett. 2012 Sep 15;22(18):5915-8. doi: 10.1016/j.bmcl.2012.07.069. Epub 2012 Jul 27. Bioorg Med Chem Lett. 2012. PMID: 22884991
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