Azuaje J - Search Results

1

Exploring the Effect of Halogenation in a Series of Potent and Selective A_2B Adenosine Receptor Antagonists.

Prieto-Díaz R, González-Gómez M, Fojo-Carballo H, Azuaje J, El Maatougui A, Majellaro M, Loza MI, Brea J, Fernández-Dueñas V, Paleo MR, Díaz-Holguín A, Garcia-Pinel B, Mallo-Abreu A, Estévez JC, Andújar-Arias A, García-Mera X, Gomez-Tourino I, Ciruela F, Salas CO, Gutiérrez-de-Terán H, Sotelo E. Prieto-Díaz R, et al. Among authors: azuaje j. J Med Chem. 2023 Jan 12;66(1):890-912. doi: 10.1021/acs.jmedchem.2c01768. Epub 2022 Dec 14. J Med Chem. 2023. PMID: 36517209 Free PMC article.

2

Silica-supported aluminum chloride-assisted solution phase synthesis of pyridazinone-based antiplatelet agents.

El Maatougui A, Azuaje J, Sotelo E, Caamaño O, Coelho A. El Maatougui A, et al. Among authors: azuaje j. ACS Comb Sci. 2011 Jan 10;13(1):7-12. doi: 10.1021/co100017h. Epub 2010 Nov 9. ACS Comb Sci. 2011. PMID: 21247118

3

Supported p-toluenesulfonic acid as a highly robust and eco-friendly isocyanide scavenger.

Azuaje J, Coelho A, Maatougui AE, Blanco JM, Sotelo E. Azuaje J, et al. ACS Comb Sci. 2011 Jan 10;13(1):89-95. doi: 10.1021/co100035z. Epub 2010 Nov 10. ACS Comb Sci. 2011. PMID: 21247131

4

Discovery and preliminary SAR of 5-arylidene-2,2-dimethyl-1,3-dioxane- 4,6-diones as platelet aggregation inhibitors.

El Maatougui A, Azuaje J, Coelho A, Cano E, Yañez M, López C, Yaziji V, Carbajales C, Sotelo E. El Maatougui A, et al. Among authors: azuaje j. Comb Chem High Throughput Screen. 2012 Aug;15(7):551-4. doi: 10.2174/138620712801619122. Comb Chem High Throughput Screen. 2012. PMID: 22272691

5

Multicomponent assembly of diverse pyrazin-2(1H)-one chemotypes.

Azuaje J, El Maatougui A, Pérez-Rubio JM, Coelho A, Fernández F, Sotelo E. Azuaje J, et al. J Org Chem. 2013 May 3;78(9):4402-9. doi: 10.1021/jo4003163. Epub 2013 Apr 12. J Org Chem. 2013. PMID: 23551216

6

Three-component assembly of structurally diverse 2-aminopyrimidine-5-carbonitriles.

Val C, Crespo A, Yaziji V, Coelho A, Azuaje J, El Maatougui A, Carbajales C, Sotelo E. Val C, et al. Among authors: azuaje j. ACS Comb Sci. 2013 Jul 8;15(7):370-8. doi: 10.1021/co4000503. Epub 2013 Jun 6. ACS Comb Sci. 2013. PMID: 23697392

7

Copper-catalyzed Huisgen 1,3-dipolar cycloaddition under oxidative conditions: polymer-assisted assembly of 4-acyl-1-substituted-1,2,3-triazoles.

Diz PM, Coelho A, El Maatougui A, Azuaje J, Caamaño O, Gil Á, Sotelo E. Diz PM, et al. Among authors: azuaje j. J Org Chem. 2013 Jul 5;78(13):6540-9. doi: 10.1021/jo400800j. Epub 2013 Jun 14. J Org Chem. 2013. PMID: 23738944

8

Ugi-based approaches to quinoxaline libraries.

Azuaje J, El Maatougui A, García-Mera X, Sotelo E. Azuaje J, et al. ACS Comb Sci. 2014 Aug 11;16(8):403-11. doi: 10.1021/co500036n. Epub 2014 May 14. ACS Comb Sci. 2014. PMID: 24800648

9

Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists.

Crespo A, El Maatougui A, Biagini P, Azuaje J, Coelho A, Brea J, Loza MI, Cadavid MI, García-Mera X, Gutiérrez-de-Terán H, Sotelo E. Crespo A, et al. Among authors: azuaje j. ACS Med Chem Lett. 2013 Oct 3;4(11):1031-6. doi: 10.1021/ml400185v. eCollection 2013 Nov 14. ACS Med Chem Lett. 2013. PMID: 24900602 Free PMC article.

10

Structure-based design of new KSP-Eg5 inhibitors assisted by a targeted multicomponent reaction.

Carbajales C, Prado MÁ, Gutiérrez-de-Terán H, Cores A, Azuaje J, Novio S, Nuñez MJ, Fernández-García B, Sotelo E, García-Mera X, Sánchez-Lazo P, Freire-Garabal M, Coelho A. Carbajales C, et al. Among authors: azuaje j. Chembiochem. 2014 Jul 7;15(10):1471-80. doi: 10.1002/cbic.201402089. Epub 2014 Jun 18. Chembiochem. 2014. PMID: 24943831

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