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Optimization of physicochemical properties of pyrrolidine GPR40 AgoPAMs results in a differentiated profile with improved pharmacokinetics and reduced off-target activities.
Bioorg Med Chem. 2023 May 1;85:117273. doi: 10.1016/j.bmc.2023.117273. Epub 2023 Apr 4.
Bioorg Med Chem. 2023.
PMID: 37030194
Synthesis and evaluation of azabicyclo[3.2.1]octane derivatives as potent mixed vasopressin antagonists.
Crombie AL, Antrilli TM, Campbell BA, Crandall DL, Failli AA, He Y, Kern JC, Moore WJ, Nogle LM, Trybulski EJ.
Crombie AL, et al. Among authors: antrilli tm.
Bioorg Med Chem Lett. 2010 Jun 15;20(12):3742-5. doi: 10.1016/j.bmcl.2010.04.068. Epub 2010 Apr 21.
Bioorg Med Chem Lett. 2010.
PMID: 20471258
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Effect of tiplaxtinin (PAI-039), an orally bioavailable PAI-1 antagonist, in a rat model of thrombosis.
Hennan JK, Morgan GA, Swillo RE, Antrilli TM, Mugford C, Vlasuk GP, Gardell SJ, Crandall DL.
Hennan JK, et al. Among authors: antrilli tm.
J Thromb Haemost. 2008 Sep;6(9):1558-64. doi: 10.1111/j.1538-7836.2008.03063.x. Epub 2008 Jul 4.
J Thromb Haemost. 2008.
PMID: 18624980
Free article.
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Synthesis and SAR of 2-carboxylic acid indoles as inhibitors of plasminogen activator inhibitor-1.
Hu B, Jetter JW, Wrobel JE, Antrilli TM, Bauer JS, Di L, Polakowski S, Jain U, Crandall DL.
Hu B, et al. Among authors: antrilli tm.
Bioorg Med Chem Lett. 2005 Aug 1;15(15):3514-8. doi: 10.1016/j.bmcl.2005.05.095.
Bioorg Med Chem Lett. 2005.
PMID: 15982877
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Evaluation of PAI-039 [{1-benzyl-5-[4-(trifluoromethoxy)phenyl]-1H-indol-3-yl}(oxo)acetic acid], a novel plasminogen activator inhibitor-1 inhibitor, in a canine model of coronary artery thrombosis.
Hennan JK, Elokdah H, Leal M, Ji A, Friedrichs GS, Morgan GA, Swillo RE, Antrilli TM, Hreha A, Crandall DL.
Hennan JK, et al. Among authors: antrilli tm.
J Pharmacol Exp Ther. 2005 Aug;314(2):710-6. doi: 10.1124/jpet.105.084129. Epub 2005 Apr 28.
J Pharmacol Exp Ther. 2005.
PMID: 15860572
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Design and synthesis of oxadiazolidinediones as inhibitors of plasminogen activator inhibitor-1.
Gopalsamy A, Kincaid SL, Ellingboe JW, Groeling TM, Antrilli TM, Krishnamurthy G, Aulabaugh A, Friedrichs GS, Crandall DL.
Gopalsamy A, et al. Among authors: antrilli tm.
Bioorg Med Chem Lett. 2004 Jul 5;14(13):3477-80. doi: 10.1016/j.bmcl.2004.04.058.
Bioorg Med Chem Lett. 2004.
PMID: 15177456
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WAY-140312 reduces plasma PAI-1 while maintaining normal platelet aggregation.
Crandall DL, Hennan JK, Elokdah H, Krishnamurthy G, Antrilli TM, Bauer JS, Morgan GA, Swillo RE.
Crandall DL, et al. Among authors: antrilli tm.
Biochem Biophys Res Commun. 2003 Nov 28;311(4):904-8. doi: 10.1016/j.bbrc.2003.10.088.
Biochem Biophys Res Commun. 2003.
PMID: 14623266
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Release of PAI-1 by human preadipocytes and adipocytes independent of insulin and IGF-1.
Crandall DL, Groeling TM, Busler DE, Antrilli TM.
Crandall DL, et al. Among authors: antrilli tm.
Biochem Biophys Res Commun. 2000 Dec 29;279(3):984-8. doi: 10.1006/bbrc.2000.4045.
Biochem Biophys Res Commun. 2000.
PMID: 11162462
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