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Year Number of Results
2014 1
2015 1
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2018 2
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2020 4
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2023 7
2024 4

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Page 1
A novel bioresponsive self-immolative spacer based on aza-quinone methide reactivity for the controlled release of thiols, phenols, amines, sulfonamides or amides.
Ermini E, Brai A, Cini E, Finetti F, Giannini G, Padula D, Paradisi L, Poggialini F, Trabalzini L, Tolu P, Taddei M. Ermini E, et al. Among authors: brai a. Chem Sci. 2024 Apr 2;15(16):6168-6177. doi: 10.1039/d4sc01576b. eCollection 2024 Apr 24. Chem Sci. 2024. PMID: 38665538 Free PMC article.
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors.
Di Stefano M, Masoni S, Bononi G, Poli G, Galati S, Gado F, Manzi S, Vagaggini C, Brai A, Caligiuri I, Asif K, Rizzolio F, Macchia M, Chicca A, Sodi A, Di Bussolo V, Minutolo F, Meier P, Gertsch J, Granchi C, Dreassi E, Tuccinardi T. Di Stefano M, et al. Among authors: brai a. Eur J Med Chem. 2024 Jan 5;263:115916. doi: 10.1016/j.ejmech.2023.115916. Epub 2023 Nov 2. Eur J Med Chem. 2024. PMID: 37976705 Free article.
Pseudorabies virus hijacks DDX3X, initiating an addictive "mad itch" and immune suppression, to facilitate viral spread.
Cronin SJF, Tejada MA, Song R, Laval K, Cikes D, Ji M, Brai A, Stadlmann J, Novatchikova M, Perlot T, Ali OH, Botta L, Decker T, Lazovic J, Hagelkruys A, Enquist L, Rao S, Koyuncu OO, Penninger JM. Cronin SJF, et al. Among authors: brai a. bioRxiv [Preprint]. 2023 May 9:2023.05.09.539956. doi: 10.1101/2023.05.09.539956. bioRxiv. 2023. PMID: 37214906 Free PMC article. Preprint.
Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme.
Poggialini F, Vagaggini C, Brai A, Pasqualini C, Crespan E, Maga G, Perini C, Cabella N, Botta L, Musumeci F, Frosini M, Schenone S, Dreassi E. Poggialini F, et al. Among authors: brai a. Pharmaceutics. 2023 Jan 30;15(2):453. doi: 10.3390/pharmaceutics15020453. Pharmaceutics. 2023. PMID: 36839775 Free PMC article.
32 results