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2,2,2-trifluoro-1-(1,4,5,6-tetrahydropyridin-3-yl)ethanone derivative as efflux pump inhibitor in Mycobacterium tuberculosis.
Halicki PCB, Vianna JS, Zanatta N, de Andrade VP, de Oliveira M, Mateus M, da Silva MV, Rodrigues V Júnior, Ramos DF, Almeida da Silva PE. Halicki PCB, et al. Among authors: almeida da silva pe. Bioorg Med Chem Lett. 2021 Jun 15;42:128088. doi: 10.1016/j.bmcl.2021.128088. Epub 2021 May 6. Bioorg Med Chem Lett. 2021. PMID: 33964440
Synthesis and in vitro antimycobacterial activity of 3-substituted 5-hydroxy-5-trifluoro[chloro]methyl-4,5-dihydro-1H-1-(isonicotinoyl) pyrazoles.
Almeida da Silva PE, Ramos DF, Bonacorso HG, de la Iglesia AI, Oliveira MR, Coelho T, Navarini J, Morbidoni HR, Zanatta N, Martins MA. Almeida da Silva PE, et al. Int J Antimicrob Agents. 2008 Aug;32(2):139-44. doi: 10.1016/j.ijantimicag.2008.03.019. Epub 2008 Jun 20. Int J Antimicrob Agents. 2008. PMID: 18571384
In vitro and in silico analysis of the efficiency of tetrahydropyridines as drug efflux inhibitors in Escherichia coli.
Silva L Jr, Carrion LL, von Groll A, Costa SS, Junqueira E, Ramos DF, Cantos J, Seus VR, Couto I, Fernandes LD, Bonacorso HG, Martins MA, Zanatta N, Viveiros M, Machado KS, Almeida da Silva PE. Silva L Jr, et al. Among authors: almeida da silva pe. Int J Antimicrob Agents. 2017 Mar;49(3):308-314. doi: 10.1016/j.ijantimicag.2016.11.024. Epub 2017 Jan 30. Int J Antimicrob Agents. 2017. PMID: 28153476 Free article.
Tetrahydropyridine derivative as efflux inhibitor in Mycobacterium abscessus.
Vianna JS, Ramis IB, Bierhals D, von Groll A, Ramos DF, Zanatta N, Lourenço MC, Viveiros M, Almeida da Silva PE. Vianna JS, et al. Among authors: almeida da silva pe. J Glob Antimicrob Resist. 2019 Jun;17:296-299. doi: 10.1016/j.jgar.2018.12.020. Epub 2019 Jan 7. J Glob Antimicrob Resist. 2019. PMID: 30630106
Design of hybrid molecules as antimycobacterial compounds: Synthesis of isoniazid-naphthoquinone derivatives and their activity against susceptible and resistant strains of Mycobacterium tuberculosis.
Reis WJ, Bozzi ÍAO, Ribeiro MF, Halicki PCB, Ferreira LA, Almeida da Silva PE, Ramos DF, de Simone CA, da Silva Júnior EN. Reis WJ, et al. Among authors: almeida da silva pe, da silva junior en. Bioorg Med Chem. 2019 Sep 15;27(18):4143-4150. doi: 10.1016/j.bmc.2019.07.045. Epub 2019 Jul 27. Bioorg Med Chem. 2019. PMID: 31378595 Free article.
Chemical Profile and Antimicrobial Activity of the Marine Diatom Chaetoceros muelleri.
Ramos DF, Bartolomeu Halicki PC, da Silva Canielles Caprara C, Borges P, da R M D'Oca C, de Fátima C Santos M, D'Oca MGM, Roselet F, Almeida da Silva PE, Abreu PC. Ramos DF, et al. Among authors: almeida da silva pe. Chem Biodivers. 2022 May;19(5):e202100846. doi: 10.1002/cbdv.202100846. Epub 2022 Mar 25. Chem Biodivers. 2022. PMID: 35290725
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