Alcaro S - Search Results

1

Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis.

Albertini C, Salerno A, Atzeni S, Uliassi E, Massenzio F, Maruca A, Rocca R, Mecava M, Silva FSG, Mena D, Valente P, Duarte AI, Chavarria D, Bissaro M, Moro S, Federico S, Spalluto G, Soukup O, Borges F, Alcaro S, Monti B, Oliveira PJ, Menéndez JC, Bolognesi ML. Albertini C, et al. Among authors: alcaro s. ACS Chem Neurosci. 2022 Aug 3;13(15):2252-2260. doi: 10.1021/acschemneuro.2c00261. Epub 2022 Jul 22. ACS Chem Neurosci. 2022. PMID: 35868251 Free PMC article.

2

Chromone-2- and -3-carboxylic acids inhibit differently monoamine oxidases A and B.

Alcaro S, Gaspar A, Ortuso F, Milhazes N, Orallo F, Uriarte E, Yáñez M, Borges F. Alcaro S, et al. Bioorg Med Chem Lett. 2010 May 1;20(9):2709-12. doi: 10.1016/j.bmcl.2010.03.081. Epub 2010 Mar 27. Bioorg Med Chem Lett. 2010. PMID: 20382016

3

Chromone, a privileged scaffold for the development of monoamine oxidase inhibitors.

Gaspar A, Silva T, Yáñez M, Vina D, Orallo F, Ortuso F, Uriarte E, Alcaro S, Borges F. Gaspar A, et al. Among authors: alcaro s. J Med Chem. 2011 Jul 28;54(14):5165-73. doi: 10.1021/jm2004267. Epub 2011 Jul 1. J Med Chem. 2011. PMID: 21696156

4

Targeting unimolecular G-quadruplex nucleic acids: a new paradigm for the drug discovery?

Parrotta L, Ortuso F, Moraca F, Rocca R, Costa G, Alcaro S, Artese A. Parrotta L, et al. Among authors: alcaro s. Expert Opin Drug Discov. 2014 Oct;9(10):1167-87. doi: 10.1517/17460441.2014.941353. Epub 2014 Aug 11. Expert Opin Drug Discov. 2014. PMID: 25109710 Review.

5

Structure-based virtual screening of novel natural alkaloid derivatives as potential binders of h-telo and c-myc DNA G-quadruplex conformations.

Rocca R, Moraca F, Costa G, Alcaro S, Distinto S, Maccioni E, Ortuso F, Artese A, Parrotta L. Rocca R, et al. Among authors: alcaro s. Molecules. 2014 Dec 24;20(1):206-23. doi: 10.3390/molecules20010206. Molecules. 2014. PMID: 25547724 Free PMC article.

6

Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress.

Aiello F, Badolato M, Pessina F, Sticozzi C, Maestrini V, Aldinucci C, Luongo L, Guida F, Ligresti A, Artese A, Allarà M, Costa G, Frosini M, Schiano Moriello A, De Petrocellis L, Valacchi G, Alcaro S, Maione S, Di Marzo V, Corelli F, Brizzi A. Aiello F, et al. Among authors: alcaro s. ACS Chem Neurosci. 2016 Jun 15;7(6):737-48. doi: 10.1021/acschemneuro.5b00333. Epub 2016 Mar 22. ACS Chem Neurosci. 2016. PMID: 26942555

7

Discovery of New Chemical Entities for Old Targets: Insights on the Lead Optimization of Chromone-Based Monoamine Oxidase B (MAO-B) Inhibitors.

Reis J, Cagide F, Chavarria D, Silva T, Fernandes C, Gaspar A, Uriarte E, Remião F, Alcaro S, Ortuso F, Borges F. Reis J, et al. Among authors: alcaro s. J Med Chem. 2016 Jun 23;59(12):5879-93. doi: 10.1021/acs.jmedchem.6b00527. Epub 2016 Jun 10. J Med Chem. 2016. PMID: 27244485

8

A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences.

Costa G, Rocca R, Moraca F, Talarico C, Romeo I, Ortuso F, Alcaro S, Artese A. Costa G, et al. Among authors: alcaro s. Mol Inform. 2016 Sep;35(8-9):391-402. doi: 10.1002/minf.201501040. Epub 2016 Jun 24. Mol Inform. 2016. PMID: 27546043

9

Identification of G-quadruplex DNA/RNA binders: Structure-based virtual screening and biophysical characterization.

Rocca R, Moraca F, Costa G, Nadai M, Scalabrin M, Talarico C, Distinto S, Maccioni E, Ortuso F, Artese A, Alcaro S, Richter SN. Rocca R, et al. Among authors: alcaro s. Biochim Biophys Acta Gen Subj. 2017 May;1861(5 Pt B):1329-1340. doi: 10.1016/j.bbagen.2016.12.023. Epub 2016 Dec 23. Biochim Biophys Acta Gen Subj. 2017. PMID: 28025082

10

Molecular recognition of a carboxy pyridostatin toward G-quadruplex structures: Why does it prefer RNA?

Rocca R, Talarico C, Moraca F, Costa G, Romeo I, Ortuso F, Alcaro S, Artese A. Rocca R, et al. Among authors: alcaro s. Chem Biol Drug Des. 2017 Nov;90(5):919-925. doi: 10.1111/cbdd.13015. Epub 2017 Jun 6. Chem Biol Drug Des. 2017. PMID: 28459507

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