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Synthesis, X-ray Structure, Hirshfeld, DFT Conformational, Cytotoxic, and Anti-Toxoplasma Studies of New Indole-Hydrazone Derivatives.
Int J Mol Sci. 2023 Aug 26;24(17):13251. doi: 10.3390/ijms241713251.
Int J Mol Sci. 2023.
PMID: 37686056
Free PMC article.
Discovery of Potent Indolyl-Hydrazones as Kinase Inhibitors for Breast Cancer: Synthesis, X-ray Single-Crystal Analysis, and In Vitro and In Vivo Anti-Cancer Activity Evaluation.
Salama EE, Youssef MF, Aboelmagd A, Boraei ATA, Nafie MS, Haukka M, Barakat A, Sarhan AAM.
Salama EE, et al.
Pharmaceuticals (Basel). 2023 Dec 13;16(12):1724. doi: 10.3390/ph16121724.
Pharmaceuticals (Basel). 2023.
PMID: 38139850
Free PMC article.
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A novel alpha-amylase inhibitor-based spirooxindole-pyrrolidine-clubbed thiochromene-pyrzaole pharmacophores: Unveiling the [3+2] cycloaddition reaction by molecular electron density theory.
Islam MS, Al-Majid AM, Haukka M, Parveen Z, Ravaiz N, Wadood A, Rehman AU, Ríos-Gutiérrez M, Domingo LR, Barakat A.
Islam MS, et al.
Chem Biol Drug Des. 2023 Nov;102(5):972-995. doi: 10.1111/cbdd.14299. Epub 2023 Aug 10.
Chem Biol Drug Des. 2023.
PMID: 37563748
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