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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
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2016 | 1 |
2018 | 3 |
2019 | 1 |
2020 | 1 |
2021 | 1 |
2024 | 0 |
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Discovery of phenylalanine derivatives as potent HIV-1 capsid inhibitors from click chemistry-based compound library.
Eur J Med Chem. 2018 Oct 5;158:478-492. doi: 10.1016/j.ejmech.2018.09.029. Epub 2018 Sep 11.
Eur J Med Chem. 2018.
PMID: 30243152
Free PMC article.
Kinetic Characterization of Novel HIV-1 Entry Inhibitors: Discovery of a Relationship between Off-Rate and Potency.
Meuser ME, Murphy MB, Rashad AA, Cocklin S.
Meuser ME, et al.
Molecules. 2018 Aug 3;23(8):1940. doi: 10.3390/molecules23081940.
Molecules. 2018.
PMID: 30081466
Free PMC article.
Item in Clipboard
Field-Based Affinity Optimization of a Novel Azabicyclohexane Scaffold HIV-1 Entry Inhibitor.
Meuser ME, Rashad AA, Ozorowski G, Dick A, Ward AB, Cocklin S.
Meuser ME, et al.
Molecules. 2019 Apr 22;24(8):1581. doi: 10.3390/molecules24081581.
Molecules. 2019.
PMID: 31013646
Free PMC article.
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Phosphorylation of the RNA-binding protein Dazl by MAPKAP kinase 2 regulates spermatogenesis.
Williams PA, Krug MS, McMillan EA, Peake JD, Davis TL, Cocklin S, Strochlic TI.
Williams PA, et al.
Mol Biol Cell. 2016 Aug 1;27(15):2341-50. doi: 10.1091/mbc.E15-11-0773. Epub 2016 Jun 8.
Mol Biol Cell. 2016.
PMID: 27280388
Free PMC article.
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Rapid Optimization of the Metabolic Stability of a Human Immunodeficiency Virus Type-1 Capsid Inhibitor Using a Multistep Computational Workflow.
Meuser ME, Reddy PAN, Dick A, Maurancy JM, Salvino JM, Cocklin S.
Meuser ME, et al.
J Med Chem. 2021 Apr 8;64(7):3747-3766. doi: 10.1021/acs.jmedchem.0c01810. Epub 2021 Mar 22.
J Med Chem. 2021.
PMID: 33750123
Free PMC article.
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Exploring Modifications of an HIV-1 Capsid Inhibitor: Design, Synthesis, and Mechanism of Action.
Xu JP, Francis AC, Meuser ME, Mankowski M, Ptak RG, Rashad AA, Melikyan GB, Cocklin S.
Xu JP, et al.
J Drug Des Res. 2018;5(2):1070. Epub 2018 Aug 13.
J Drug Des Res. 2018.
PMID: 30393786
Free PMC article.
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Composition and Orientation of the Core Region of Novel HIV-1 Entry Inhibitors Influences Metabolic Stability.
Karadsheh R, Meuser ME, Cocklin S.
Karadsheh R, et al.
Molecules. 2020 Mar 21;25(6):1430. doi: 10.3390/molecules25061430.
Molecules. 2020.
PMID: 32245167
Free PMC article.
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