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Synthesis and pharmacological validation of a novel radioligand for the orphan GPR88 receptor.
Bioorg Med Chem Lett. 2023 Jan 15;80:129120. doi: 10.1016/j.bmcl.2022.129120. Epub 2022 Dec 29.
Bioorg Med Chem Lett. 2023.
PMID: 36587872
Free PMC article.
Evaluation of Amide Bioisosteres Leading to 1,2,3-Triazole Containing Compounds as GPR88 Agonists: Design, Synthesis, and Structure-Activity Relationship Studies.
Rahman MT, Decker AM, Laudermilk L, Maitra R, Ma W, Ben Hamida S, Darcq E, Kieffer BL, Jin C.
Rahman MT, et al.
J Med Chem. 2021 Aug 26;64(16):12397-12413. doi: 10.1021/acs.jmedchem.1c01075. Epub 2021 Aug 13.
J Med Chem. 2021.
PMID: 34387471
Free PMC article.
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