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Screening for dimethylarginine dimethylaminohydrolase inhibitors reveals ebselen as a bioavailable inactivator.
ACS Med Chem Lett. 2011;2(8):592-596. doi: 10.1021/ml2000824.
ACS Med Chem Lett. 2011.
PMID: 21927644
Free PMC article.
On the mechanism of dimethylarginine dimethylaminohydrolase inactivation by 4-halopyridines.
Johnson CM, Monzingo AF, Ke Z, Yoon DW, Linsky TW, Guo H, Robertus JD, Fast W.
Johnson CM, et al.
J Am Chem Soc. 2011 Jul 20;133(28):10951-9. doi: 10.1021/ja2033684. Epub 2011 Jun 23.
J Am Chem Soc. 2011.
PMID: 21630706
Free PMC article.
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Discovery of peptidylarginine deiminase-4 substrates by protein array: antagonistic citrullination and methylation of human ribosomal protein S2.
Guo Q, Bedford MT, Fast W.
Guo Q, et al.
Mol Biosyst. 2011 Jul;7(7):2286-95. doi: 10.1039/c1mb05089c. Epub 2011 May 16.
Mol Biosyst. 2011.
PMID: 21584310
Free PMC article.
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A continuous, fluorescent, high-throughput assay for human dimethylarginine dimethylaminohydrolase-1.
Linsky T, Fast W.
Linsky T, et al.
J Biomol Screen. 2011 Oct;16(9):1089-97. doi: 10.1177/1087057111417712. Epub 2011 Sep 15.
J Biomol Screen. 2011.
PMID: 21921133
Free PMC article.
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