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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
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2020 | 1 |
2021 | 1 |
2022 | 2 |
2023 | 3 |
2024 | 2 |
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Page 1
Targeting the relaxin-3/RXFP3 system: a patent review for the last two decades.
Expert Opin Ther Pat. 2024 Jan-Feb;34(1-2):71-81. doi: 10.1080/13543776.2024.2338099. Epub 2024 Apr 4.
Expert Opin Ther Pat. 2024.
PMID: 38573177
Review.
The GPR88 agonist RTI-13951-33 reduces alcohol drinking and seeking in mice.
Ben Hamida S, Carter M, Darcq E, Sourty M, Rahman MT, Decker AM, Jin C, Kieffer BL.
Ben Hamida S, et al.
Addict Biol. 2022 Nov;27(6):e13227. doi: 10.1111/adb.13227.
Addict Biol. 2022.
PMID: 36301207
Free PMC article.
Item in Clipboard
Synthesis and pharmacological validation of a novel radioligand for the orphan GPR88 receptor.
Decker AM, Rahman MT, Kormos CM, Hesk D, Darcq E, Kieffer BL, Jin C.
Decker AM, et al.
Bioorg Med Chem Lett. 2023 Jan 15;80:129120. doi: 10.1016/j.bmcl.2022.129120. Epub 2022 Dec 29.
Bioorg Med Chem Lett. 2023.
PMID: 36587872
Free PMC article.
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Design, Synthesis, and Structure-Activity Relationship Studies of (4-Alkoxyphenyl)glycinamides and Bioisosteric 1,3,4-Oxadiazoles as GPR88 Agonists.
Rahman MT, Decker AM, Langston TL, Mathews KM, Laudermilk L, Maitra R, Ma W, Darcq E, Kieffer BL, Jin C.
Rahman MT, et al.
J Med Chem. 2020 Dec 10;63(23):14989-15012. doi: 10.1021/acs.jmedchem.0c01581. Epub 2020 Nov 18.
J Med Chem. 2020.
PMID: 33205975
Free PMC article.
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Improvement of the Metabolic Stability of GPR88 Agonist RTI-13951-33: Design, Synthesis, and Biological Evaluation.
Rahman MT, Decker AM, Ben Hamida S, Perrey DA, Chaminda Lakmal HH, Maitra R, Darcq E, Kieffer BL, Jin C.
Rahman MT, et al.
J Med Chem. 2023 Feb 23;66(4):2964-2978. doi: 10.1021/acs.jmedchem.2c01983. Epub 2023 Feb 7.
J Med Chem. 2023.
PMID: 36749855
Free PMC article.
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Evaluation of Amide Bioisosteres Leading to 1,2,3-Triazole Containing Compounds as GPR88 Agonists: Design, Synthesis, and Structure-Activity Relationship Studies.
Rahman MT, Decker AM, Laudermilk L, Maitra R, Ma W, Ben Hamida S, Darcq E, Kieffer BL, Jin C.
Rahman MT, et al.
J Med Chem. 2021 Aug 26;64(16):12397-12413. doi: 10.1021/acs.jmedchem.1c01075. Epub 2021 Aug 13.
J Med Chem. 2021.
PMID: 34387471
Free PMC article.
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Design, Synthesis, and Structure-Activity Relationship Studies of Novel GPR88 Agonists (4-Substituted-phenyl)acetamides Based on the Reversed Amide Scaffold.
Rahman MT, Guan D, Chaminda Lakmal HH, Decker AM, Imler GH, Kerr AT, Harris DL, Jin C.
Rahman MT, et al.
ACS Chem Neurosci. 2024 Jan 3;15(1):169-192. doi: 10.1021/acschemneuro.3c00684. Epub 2023 Dec 12.
ACS Chem Neurosci. 2024.
PMID: 38086012
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