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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
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2019 | 1 |
2020 | 1 |
2021 | 1 |
2023 | 3 |
2024 | 0 |
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6 results
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Page 1
Small-molecule tools for YEATS domain proteins.
Curr Opin Chem Biol. 2023 Dec;77:102404. doi: 10.1016/j.cbpa.2023.102404. Epub 2023 Nov 3.
Curr Opin Chem Biol. 2023.
PMID: 37924571
Review.
Acetyl-CoA biosynthesis drives resistance to histone acetyltransferase inhibition.
Bishop TR, Subramanian C, Bilotta EM, Garnar-Wortzel L, Ramos AR, Zhang Y, Asiaban JN, Ott CJ, Rock CO, Erb MA.
Bishop TR, et al.
Nat Chem Biol. 2023 Oct;19(10):1215-1222. doi: 10.1038/s41589-023-01320-7. Epub 2023 May 1.
Nat Chem Biol. 2023.
PMID: 37127754
Free PMC article.
Item in Clipboard
Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities.
Zhang Y, Remillard D, Onubogu U, Karakyriakou B, Asiaban JN, Ramos AR, Bowland K, Bishop TR, Barta PA, Nance S, Durbin AD, Ott CJ, Janiszewska M, Cravatt BF, Erb MA.
Zhang Y, et al.
Nat Struct Mol Biol. 2023 Aug;30(8):1160-1171. doi: 10.1038/s41594-023-01041-4. Epub 2023 Jul 24.
Nat Struct Mol Biol. 2023.
PMID: 37488358
Free PMC article.
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Pharmacological Modulation of Transcriptional Coregulators in Cancer.
Bishop TR, Zhang Y, Erb MA.
Bishop TR, et al.
Trends Pharmacol Sci. 2019 Jun;40(6):388-402. doi: 10.1016/j.tips.2019.04.004. Epub 2019 May 8.
Trends Pharmacol Sci. 2019.
PMID: 31078321
Free PMC article.
Review.
Item in Clipboard
Chemical Inhibition of ENL/AF9 YEATS Domains in Acute Leukemia.
Garnar-Wortzel L, Bishop TR, Kitamura S, Milosevich N, Asiaban JN, Zhang X, Zheng Q, Chen E, Ramos AR, Ackerman CJ, Hampton EN, Chatterjee AK, Young TS, Hull MV, Sharpless KB, Cravatt BF, Wolan DW, Erb MA.
Garnar-Wortzel L, et al.
ACS Cent Sci. 2021 May 26;7(5):815-830. doi: 10.1021/acscentsci.0c01550. Epub 2021 Apr 30.
ACS Cent Sci. 2021.
PMID: 34079898
Free PMC article.
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Cell-Based Ligand Discovery for the ENL YEATS Domain.
Asiaban JN, Milosevich N, Chen E, Bishop TR, Wang J, Zhang Y, Ackerman CJ, Hampton EN, Young TS, Hull MV, Cravatt BF, Erb MA.
Asiaban JN, et al.
ACS Chem Biol. 2020 Apr 17;15(4):895-903. doi: 10.1021/acschembio.0c00124. Epub 2020 Mar 19.
ACS Chem Biol. 2020.
PMID: 32176478
Free PMC article.
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