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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
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2011 | 1 |
2012 | 1 |
2020 | 1 |
2024 | 0 |
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Nek7 conformational flexibility and inhibitor binding probed through protein engineering of the R-spine.
Biochem J. 2020 Apr 30;477(8):1525-1539. doi: 10.1042/BCJ20200128.
Biochem J. 2020.
PMID: 32242624
Free PMC article.
Benzimidazole inhibitors induce a DFG-out conformation of never in mitosis gene A-related kinase 2 (Nek2) without binding to the back pocket and reveal a nonlinear structure-activity relationship.
Solanki S, Innocenti P, Mas-Droux C, Boxall K, Barillari C, van Montfort RL, Aherne GW, Bayliss R, Hoelder S.
Solanki S, et al.
J Med Chem. 2011 Mar 24;54(6):1626-39. doi: 10.1021/jm1011726. Epub 2011 Mar 2.
J Med Chem. 2011.
PMID: 21366329
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Design of potent and selective hybrid inhibitors of the mitotic kinase Nek2: structure-activity relationship, structural biology, and cellular activity.
Innocenti P, Cheung KM, Solanki S, Mas-Droux C, Rowan F, Yeoh S, Boxall K, Westlake M, Pickard L, Hardy T, Baxter JE, Aherne GW, Bayliss R, Fry AM, Hoelder S.
Innocenti P, et al.
J Med Chem. 2012 Apr 12;55(7):3228-41. doi: 10.1021/jm201683b. Epub 2012 Mar 23.
J Med Chem. 2012.
PMID: 22404346
Free PMC article.
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