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Rolapitant Is a Reversible Inhibitor of CYP2D6.
Drug Metab Dispos. 2019 Jun;47(6):567-573. doi: 10.1124/dmd.118.085928. Epub 2019 Apr 5.
Drug Metab Dispos. 2019.
PMID: 30952677
Free PMC article.
Metoclopramide is metabolized by CYP2D6 and is a reversible inhibitor, but not inactivator, of CYP2D6.
Livezey MR, Briggs ED, Bolles AK, Nagy LD, Fujiwara R, Furge LL.
Livezey MR, et al.
Xenobiotica. 2014 Apr;44(4):309-319. doi: 10.3109/00498254.2013.835885. Epub 2013 Sep 6.
Xenobiotica. 2014.
PMID: 24010633
Free PMC article.
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Mechanism-based inactivation of human cytochrome P450 3A4 by two piperazine-containing compounds.
Bolles AK, Fujiwara R, Briggs ED, Nomeir AA, Furge LL.
Bolles AK, et al.
Drug Metab Dispos. 2014 Dec;42(12):2087-96. doi: 10.1124/dmd.114.060459. Epub 2014 Oct 1.
Drug Metab Dispos. 2014.
PMID: 25273356
Free PMC article.
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Substituted imidazole of 5-fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates cytochrome P450 2D6 by protein adduction.
Nagy LD, Mocny CS, Diffenderfer LE, Hsi DJ, Butler BF, Arthur EJ, Fletke KJ, Palamanda JR, Nomeir AA, Furge LL.
Nagy LD, et al.
Drug Metab Dispos. 2011 Jun;39(6):974-83. doi: 10.1124/dmd.110.037630. Epub 2011 Mar 21.
Drug Metab Dispos. 2011.
PMID: 21422192
Free PMC article.
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Molecular analysis and modeling of inactivation of human CYP2D6 by four mechanism based inactivators.
Livezey M, Nagy LD, Diffenderfer LE, Arthur EJ, Hsi DJ, Holton JM, Furge LL.
Livezey M, et al.
Drug Metab Lett. 2012 Mar;6(1):7-14. doi: 10.2174/187231212800229318.
Drug Metab Lett. 2012.
PMID: 22372551
Free PMC article.
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