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Page 1
Polyfluoroalkylated antipyrines in Pd-catalyzed transformations.
Shchegolkov EV, Burgart YV, Matsneva DA, Borisevich SS, Kadyrova RA, Orshanskaya IR, Zarubaev VV, Saloutin VI. Shchegolkov EV, et al. Among authors: saloutin vi. RSC Adv. 2021 Oct 31;11(56):35174-35181. doi: 10.1039/d1ra06967e. eCollection 2021 Oct 28. RSC Adv. 2021. PMID: 35493195 Free PMC article.
Powerful Potential of Polyfluoroalkyl-Containing 4-Arylhydrazinylidenepyrazol-3-ones for Pharmaceuticals.
Burgart YV, Elkina NA, Shchegolkov EV, Krasnykh OP, Makhaeva GF, Triandafilova GA, Solodnikov SY, Boltneva NP, Rudakova EV, Kovaleva NV, Serebryakova OG, Ulitko MV, Borisevich SS, Gerasimova NA, Evstigneeva NP, Kozlov SA, Korolkova YV, Minin AS, Belousova AV, Mozhaitsev ES, Klabukov AM, Saloutin VI. Burgart YV, et al. Among authors: saloutin vi. Molecules. 2022 Dec 21;28(1):59. doi: 10.3390/molecules28010059. Molecules. 2022. PMID: 36615256 Free PMC article.
Conjugates of Tacrine with Salicylamide as Promising Multitarget Agents for Alzheimer's Disease.
Grishchenko MV, Makhaeva GF, Burgart YV, Rudakova EV, Boltneva NP, Kovaleva NV, Serebryakova OG, Lushchekina SV, Astakhova TY, Zhilina EF, Shchegolkov EV, Richardson RJ, Saloutin VI. Grishchenko MV, et al. Among authors: saloutin vi. ChemMedChem. 2022 May 18;17(10):e202200080. doi: 10.1002/cmdc.202200080. Epub 2022 Mar 23. ChemMedChem. 2022. PMID: 35322571 Free PMC article.
Synthesis of 4-Aminopyrazol-5-ols as Edaravone Analogs and Their Antioxidant Activity.
Burgart YV, Makhaeva GF, Krasnykh OP, Borisevich SS, Agafonova NA, Kovaleva NV, Boltneva NP, Rudakova EV, Shchegolkov EV, Triandafilova GA, Gazizov DA, Serebryakova OG, Ulitko MV, Khursan SL, Saloutin VI, Richardson RJ. Burgart YV, et al. Among authors: saloutin vi. Molecules. 2022 Nov 9;27(22):7722. doi: 10.3390/molecules27227722. Molecules. 2022. PMID: 36431823 Free PMC article.
5-Alkoxy-1-aryl-3-polyfluoroalkylpyrazoles with Antinociceptive Activity: Partial Agonists of TRPV1 Ion Channels.
Khudina OG, Burgart YV, Malkova NA, Shchegolkov EV, Krasnykh OP, Triandafilova GA, Malysheva KO, Solodnikov SY, Dubodel ES, Korolkova YV, Kozlov SA, Borisevich SS, Mozhaitsev ES, Saloutin VI. Khudina OG, et al. Among authors: saloutin vi. ChemMedChem. 2023 Jun 15;18(12):e202300063. doi: 10.1002/cmdc.202300063. Epub 2023 Apr 17. ChemMedChem. 2023. PMID: 37006199
New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones.
Elkina NA, Grishchenko MV, Shchegolkov EV, Makhaeva GF, Kovaleva NV, Rudakova EV, Boltneva NP, Lushchekina SV, Astakhova TY, Radchenko EV, Palyulin VA, Zhilina EF, Perminova AN, Lapshin LS, Burgart YV, Saloutin VI, Richardson RJ. Elkina NA, et al. Among authors: saloutin vi. Biomolecules. 2022 Oct 24;12(11):1551. doi: 10.3390/biom12111551. Biomolecules. 2022. PMID: 36358901 Free PMC article.
Novel potent bifunctional carboxylesterase inhibitors based on a polyfluoroalkyl-2-imino-1,3-dione scaffold.
Makhaeva GF, Lushchekina SV, Boltneva NP, Serebryakova OG, Kovaleva NV, Rudakova EV, Elkina NA, Shchegolkov EV, Burgart YV, Stupina TS, Terentiev AA, Radchenko EV, Palyulin VA, Saloutin VI, Bachurin SO, Richardson RJ. Makhaeva GF, et al. Among authors: saloutin vi. Eur J Med Chem. 2021 Jun 5;218:113385. doi: 10.1016/j.ejmech.2021.113385. Epub 2021 Mar 15. Eur J Med Chem. 2021. PMID: 33831780
New heteroanalogs of tricyclic ascidian alkaloids: synthesis and biological activity.
Goryaeva MV, Kushch SO, Burgart YV, Ezhikova MA, Kodess MI, Slepukhin PA, Triandafilova GA, Krasnykh OP, Yakovleva EI, Zarubaev VV, Sinegubova EO, Esaulkova IL, Shtro AA, Galochkina AV, Nikolaeva YV, Saloutin VI. Goryaeva MV, et al. Among authors: saloutin vi. Org Biomol Chem. 2021 Nov 25;19(45):9925-9935. doi: 10.1039/d1ob01843d. Org Biomol Chem. 2021. PMID: 34735561
22 results