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Page 1
6-Substituted quinolines as RORγt inverse agonists.
Bioorg Med Chem Lett. 2017 Dec 1;27(23):5277-5283. doi: 10.1016/j.bmcl.2017.10.027. Epub 2017 Oct 16.
Bioorg Med Chem Lett. 2017.
PMID: 29079472
Systems Biology and Peptide Engineering to Overcome Absorption Barriers for Oral Peptide Delivery: Dosage Form Optimization Case Study Preceding Clinical Translation.
Tyagi P, Patel C, Gibson K, MacDougall F, Pechenov SY, Will S, Revell J, Huang Y, Rosenbaum AI, Balic K, Maharoof U, Grimsby J, Subramony JA.
Tyagi P, et al. Among authors: maharoof u.
Pharmaceutics. 2023 Oct 9;15(10):2436. doi: 10.3390/pharmaceutics15102436.
Pharmaceutics. 2023.
PMID: 37896196
Free PMC article.
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(6,7-Dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenylamines: platelet-derived growth factor receptor tyrosine kinase inhibitors with broad antiproliferative activity against tumor cells.
Ho CY, Ludovici DW, Maharoof US, Mei J, Sechler JL, Tuman RW, Strobel ED, Andraka L, Yen HK, Leo G, Li J, Almond H, Lu H, DeVine A, Tominovich RM, Baker J, Emanuel S, Gruninger RH, Middleton SA, Johnson DL, Galemmo RA Jr.
Ho CY, et al. Among authors: maharoof us.
J Med Chem. 2005 Dec 29;48(26):8163-73. doi: 10.1021/jm050680m.
J Med Chem. 2005.
PMID: 16366598
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Identification and structure activity relationships of quinoline tertiary alcohol modulators of RORγt.
Kummer DA, Cummings MD, Abad M, Barbay J, Castro G, Wolin R, Kreutter KD, Maharoof U, Milligan C, Nishimura R, Pierce J, Schalk-Hihi C, Spurlino J, Urbanski M, Venkatesan H, Wang A, Woods C, Xue X, Edwards JP, Fourie AM, Leonard K.
Kummer DA, et al. Among authors: maharoof u.
Bioorg Med Chem Lett. 2017 May 1;27(9):2047-2057. doi: 10.1016/j.bmcl.2017.02.044. Epub 2017 Feb 21.
Bioorg Med Chem Lett. 2017.
PMID: 28318945
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Diverging stereochemical pathways in an intramolecular Diels-Alder reaction determined by dienophile structure.
Kim K, Maharoof US, Raushel J, Sulikowski GA.
Kim K, et al. Among authors: maharoof us.
Org Lett. 2003 Aug 7;5(16):2777-80. doi: 10.1021/ol034823f.
Org Lett. 2003.
PMID: 12889872
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