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Page 1
NorA, Tet(K), MepA, and MsrA Efflux Pumps in Staphylococcus aureus, their Inhibitors and 1,8-Naphthyridine Sulfonamides.
de Morais Oliveira-Tintino CD, Muniz DF, Dos Santos Barbosa CR, Silva Pereira RL, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Lacowicz Krautler MI, Barros Oliveira CV, Pereira PS, Rodrigues Teixeira AM, Tintino SR, de Menezes IRA, Melo Coutinho HD, da Silva TG. de Morais Oliveira-Tintino CD, et al. Curr Pharm Des. 2023;29(5):323-355. doi: 10.2174/1381612829666221212101501. Curr Pharm Des. 2023. PMID: 36515045 Review.
The 1,8-naphthyridines sulfonamides are NorA efflux pump inhibitors.
Oliveira-Tintino CDM, Muniz DF, Barbosa CRDS, Pereira RLS, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Pereira PS, Costa JGMD, Rodrigues FFG, Teixeira AMR, Ribeiro-Filho J, Tintino SR, de Menezes IRA, Coutinho HDM, Silva TGD. Oliveira-Tintino CDM, et al. J Glob Antimicrob Resist. 2021 Mar;24:233-240. doi: 10.1016/j.jgar.2020.11.027. Epub 2020 Dec 29. J Glob Antimicrob Resist. 2021. PMID: 33385589 Free article.
Enhancement of Antibiotic Activity by 1,8-Naphthyridine Derivatives against Multi-Resistant Bacterial Strains.
Araújo-Neto JB, Silva MMCD, Oliveira-Tintino CDM, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Ribeiro-Filho J, Siyadatpanah A, Wilairatana P, Coutinho HDM, Tintino SR. Araújo-Neto JB, et al. Among authors: mireski sl. Molecules. 2021 Dec 6;26(23):7400. doi: 10.3390/molecules26237400. Molecules. 2021. PMID: 34885981 Free PMC article.
Chemical synthesis, molecular docking and MepA efflux pump inhibitory effect by 1,8-naphthyridines sulfonamides.
Oliveira-Tintino CDM, Tintino SR, Muniz DF, Rodrigues Dos Santos Barbosa C, Pereira RLS, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Krautler MIL, Pereira PS, Balbino TCL, da Costa JGM, Rodrigues FFG, Teixeira AMR, Barreto HM, de Menezes IRA, Coutinho HDM, da Silva TG. Oliveira-Tintino CDM, et al. Eur J Pharm Sci. 2021 May 1;160:105753. doi: 10.1016/j.ejps.2021.105753. Epub 2021 Feb 10. Eur J Pharm Sci. 2021. PMID: 33581258
Efflux Pump (QacA, QacB, and QacC) and β-Lactamase Inhibitors? An Evaluation of 1,8-Naphthyridines against Staphylococcus aureus Strains.
Oliveira-Tintino CDM, Tintino SR, Justino de Araújo AC, Dos Santos Barbosa CR, Ramos Freitas P, Araújo Neto JB, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Barreto HM, Ribeiro-Filho J, de Menezes IRA, Coutinho HDM. Oliveira-Tintino CDM, et al. Molecules. 2023 Feb 15;28(4):1819. doi: 10.3390/molecules28041819. Molecules. 2023. PMID: 36838807 Free PMC article.
Do 1,8-naphthyridine sulfonamides possess an inhibitory action against Tet(K) and MsrA efflux pumps in multiresistant Staphylococcus aureus strains?
Oliveira-Tintino CDM, Tintino SR, Muniz DF, Barbosa CRDS, Pereira RLS, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Lacowicz Krautler MI, Pereira PS, Teixeira AMR, de Menezes IRA, Coutinho HDM, Silva TGD. Oliveira-Tintino CDM, et al. Microb Pathog. 2020 Oct;147:104268. doi: 10.1016/j.micpath.2020.104268. Epub 2020 Jun 20. Microb Pathog. 2020. PMID: 32574783
Potentiation of Antibiotic Activity by a Meldrum's Acid Arylamino Methylene Derivative against Multidrug-Resistant Bacterial Strains.
da Silva MMC, de Araújo-Neto JB, de Araújo ACJ, Freitas PR, de M Oliveira-Tintino CD, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Krautler MIL, Ribeiro-Filho J, Coutinho HDM, Tintino SR. da Silva MMC, et al. Among authors: mireski sl. Indian J Microbiol. 2021 Mar;61(1):100-103. doi: 10.1007/s12088-020-00910-6. Epub 2020 Oct 10. Indian J Microbiol. 2021. PMID: 33505100 Free PMC article.