Pierre Regenass - Search Results

Year	Number of Results
2014	1
2015	1
2016	2
2017	2
2018	1
2020	1
2021	1
2023	1
2024	0

1

A novel pan-selective bromodomain inhibitor for epigenetic drug design.

Warstat R, Pervaiz M, Regenass P, Amann M, Schmidtkunz K, Einsle O, Jung M, Breit B, Hügle M, Günther S. Warstat R, et al. Among authors: regenass p. Eur J Med Chem. 2023 Mar 5;249:115139. doi: 10.1016/j.ejmech.2023.115139. Epub 2023 Jan 25. Eur J Med Chem. 2023. PMID: 36736153

2

Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles.

Hügle M, Lucas X, Ostrovskyi D, Regenass P, Gerhardt S, Einsle O, Hau M, Jung M, Breit B, Günther S, Wohlwend D. Hügle M, et al. Among authors: regenass p. Angew Chem Int Ed Engl. 2017 Oct 2;56(41):12476-12480. doi: 10.1002/anie.201705516. Epub 2017 Sep 7. Angew Chem Int Ed Engl. 2017. PMID: 28766825

3

4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors Address BETi Insensitive Human Cancer Cell Lines.

Hügle M, Regenass P, Warstat R, Hau M, Schmidtkunz K, Lucas X, Wohlwend D, Einsle O, Jung M, Breit B, Günther S. Hügle M, et al. Among authors: regenass p. J Med Chem. 2020 Dec 24;63(24):15603-15620. doi: 10.1021/acs.jmedchem.0c00478. Epub 2020 Dec 4. J Med Chem. 2020. PMID: 33275431

4

Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors.

Luise C, Robaa D, Regenass P, Maurer D, Ostrovskyi D, Seifert L, Bacher J, Burgahn T, Wagner T, Seitz J, Greschik H, Park KS, Xiong Y, Jin J, Schüle R, Breit B, Jung M, Sippl W. Luise C, et al. Among authors: regenass p. Int J Mol Sci. 2021 May 31;22(11):5910. doi: 10.3390/ijms22115910. Int J Mol Sci. 2021. PMID: 34072837 Free PMC article.

5

Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia.

Regenass P, Abboud D, Daubeuf F, Lehalle C, Gizzi P, Riché S, Hachet-Haas M, Rohmer F, Gasparik V, Boeglin D, Haiech J, Knehans T, Rognan D, Heissler D, Marsol C, Villa P, Galzi JL, Hibert M, Frossard N, Bonnet D. Regenass P, et al. J Med Chem. 2018 Sep 13;61(17):7671-7686. doi: 10.1021/acs.jmedchem.8b00657. Epub 2018 Aug 28. J Med Chem. 2018. PMID: 30106292

6

Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines.

Regenass P, Bosc D, Riché S, Gizzi P, Hibert M, Karmazin L, Ganesan A, Bonnet D. Regenass P, et al. J Org Chem. 2017 Mar 17;82(6):3239-3244. doi: 10.1021/acs.joc.6b02895. Epub 2017 Mar 8. J Org Chem. 2017. PMID: 28230990

7

Convenient Access to Fluorescent Probes by Chemoselective Acylation of Hydrazinopeptides: Application to the Synthesis of the First Far-Red Ligand for Apelin Receptor Imaging.

Margathe JF, Iturrioz X, Regenass P, Karpenko IA, Humbert N, de Rocquigny H, Hibert M, Llorens-Cortes C, Bonnet D. Margathe JF, et al. Among authors: regenass p. Chemistry. 2016 Jan 22;22(4):1399-405. doi: 10.1002/chem.201503630. Epub 2015 Dec 18. Chemistry. 2016. PMID: 26682530

8

Diastereoselective synthesis of novel aza-diketopiperazines via a domino cyclohydrocarbonylation/addition process.

Regenass P, Margathe JF, Mann A, Suffert J, Hibert M, Girard N, Bonnet D. Regenass P, et al. Chem Commun (Camb). 2014 Sep 4;50(68):9657-60. doi: 10.1039/c4cc03660c. Chem Commun (Camb). 2014. PMID: 25019687

9

A step-economical multicomponent synthesis of 3D-shaped aza-diketopiperazines and their drug-like chemical space analysis.

Regenass P, Riché S, Péron F, Rognan D, Hibert M, Girard N, Bonnet D. Regenass P, et al. Org Biomol Chem. 2016 Sep 21;14(37):8859-8863. doi: 10.1039/c6ob01434h. Org Biomol Chem. 2016. PMID: 27722636

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