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Page 1
Antibiotic class with potent in vivo activity targeting lipopolysaccharide synthesis in Gram-negative bacteria.
Proc Natl Acad Sci U S A. 2024 Apr 9;121(15):e2317274121. doi: 10.1073/pnas.2317274121. Epub 2024 Apr 5.
Proc Natl Acad Sci U S A. 2024.
PMID: 38579010
Free PMC article.
Small-Molecule Inhibitors of the m7G-RNA Writer METTL1.
Nai F, Flores Espinoza MP, Invernizzi A, Vargas-Rosales PA, Bobileva O, Herok M, Caflisch A.
Nai F, et al. Among authors: bobileva o.
ACS Bio Med Chem Au. 2023 Dec 12;4(2):100-110. doi: 10.1021/acsbiomedchemau.3c00030. eCollection 2024 Apr 17.
ACS Bio Med Chem Au. 2023.
PMID: 38645929
Free PMC article.
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Synthesis and evaluation of (E)-2-(5-phenylpent-2-en-4-ynamido)cyclohex-1-ene-1-carboxylate derivatives as HCA2 receptor agonists.
Bobileva O, Ikaunieks M, Duburs G, Mandrika I, Petrovska R, Klovins J, Loza E.
Bobileva O, et al.
Bioorg Med Chem. 2017 Aug 15;25(16):4314-4329. doi: 10.1016/j.bmc.2017.06.028. Epub 2017 Jun 21.
Bioorg Med Chem. 2017.
PMID: 28668361
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3-(Adenosylthio)benzoic Acid Derivatives as SARS-CoV-2 Nsp14 Methyltransferase Inhibitors.
Bobileva O, Bobrovs R, Sirma EE, Kanepe I, Bula AL, Patetko L, Ramata-Stunda A, Grinberga S, Jirgensons A, Jaudzems K.
Bobileva O, et al.
Molecules. 2023 Jan 12;28(2):768. doi: 10.3390/molecules28020768.
Molecules. 2023.
PMID: 36677825
Free PMC article.
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Potent SARS-CoV-2 mRNA Cap Methyltransferase Inhibitors by Bioisosteric Replacement of Methionine in SAM Cosubstrate.
Bobiļeva O, Bobrovs R, Kaņepe I, Patetko L, Kalniņš G, Šišovs M, Bula AL, Gri Nberga S, Borodušķis MR, Ramata-Stunda A, Rostoks N, Jirgensons A, Ta Rs K, Jaudzems K.
Bobiļeva O, et al.
ACS Med Chem Lett. 2021 Jun 9;12(7):1102-1107. doi: 10.1021/acsmedchemlett.1c00140. eCollection 2021 Jul 8.
ACS Med Chem Lett. 2021.
PMID: 34257831
Free PMC article.
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Synthesis and evaluation of (E)-2-(acrylamido)cyclohex-1-enecarboxylic acid derivatives as HCA1, HCA2, and HCA3 receptor agonists.
Bobileva O, Bokaldere R, Gailite V, Kaula I, Ikaunieks M, Duburs G, Petrovska R, Mandrika I, Klovins J, Loza E.
Bobileva O, et al.
Bioorg Med Chem. 2014 Jul 15;22(14):3654-69. doi: 10.1016/j.bmc.2014.05.011. Epub 2014 May 17.
Bioorg Med Chem. 2014.
PMID: 24864041
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