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Page 1
Anticancer Activity of Triazolo-Thiadiazole Derivatives and Inhibition of AKT1 and AKT2 Activation.
Pharmaceutics. 2021 Apr 5;13(4):493. doi: 10.3390/pharmaceutics13040493.
Pharmaceutics. 2021.
PMID: 33916378
Free PMC article.
3,6-Disubstituted 1,2,4-Triazolo[3,4-b]Thiadiazoles with Anticancer Activity Targeting Topoisomerase II Alpha.
Sagredou S, Dalezis P, Nikoleousakos N, Nikolaou M, Voura M, Almpanakis K, Panayiotidis MI, Sarli V, Trafalis DT.
Sagredou S, et al. Among authors: nikoleousakos n.
Onco Targets Ther. 2020 Jul 28;13:7369-7386. doi: 10.2147/OTT.S254856. eCollection 2020.
Onco Targets Ther. 2020.
PMID: 32801761
Free PMC article.
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Synthesis and evaluation of new steroidal lactam conjugates with aniline mustards as potential antileukemic therapeutics.
Trafalis D, Geromichalou E, Dalezis P, Nikoleousakos N, Sarli V.
Trafalis D, et al. Among authors: nikoleousakos n.
Steroids. 2016 Nov;115:1-8. doi: 10.1016/j.steroids.2016.07.009. Epub 2016 Jul 26.
Steroids. 2016.
PMID: 27473822
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Azasteroid Alkylators as Dual Inhibitors of AKT and ERK Signaling for the Treatment of Ovarian Carcinoma.
Dalezis P, Geromichalou E, Polonifi A, Sagredou S, Nikoleousakos N, Nikolaou M, Sarli V, Panayiotidis MI, Trafalis DT.
Dalezis P, et al. Among authors: nikoleousakos n.
Cancers (Basel). 2020 May 16;12(5):1263. doi: 10.3390/cancers12051263.
Cancers (Basel). 2020.
PMID: 32429466
Free PMC article.
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Targeting on poly(ADP-ribose) polymerase activity with DNA-damaging hybrid lactam-steroid alkylators in wild-type and BRCA1-mutated ovarian cancer cells.
Trafalis DT, Polonifi A, Dalezis P, Nikoleousakos N, Katsamakas S, Sarli V.
Trafalis DT, et al. Among authors: nikoleousakos n.
Chem Biol Drug Des. 2017 Nov;90(5):854-866. doi: 10.1111/cbdd.13006. Epub 2017 May 26.
Chem Biol Drug Des. 2017.
PMID: 28432813
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The σ-hole phenomenon of halogen atoms forms the structural basis of the strong inhibitory potency of C5 halogen substituted glucopyranosyl nucleosides towards glycogen phosphorylase b.
Kantsadi AL, Hayes JM, Manta S, Skamnaki VT, Kiritsis C, Psarra AM, Koutsogiannis Z, Dimopoulou A, Theofanous S, Nikoleousakos N, Zoumpoulakis P, Kontou M, Papadopoulos G, Zographos SE, Komiotis D, Leonidas DD.
Kantsadi AL, et al. Among authors: nikoleousakos n.
ChemMedChem. 2012 Apr;7(4):722-32. doi: 10.1002/cmdc.201100533. Epub 2012 Jan 20.
ChemMedChem. 2012.
PMID: 22267166
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Cytocidal Antitumor Effects against Human Ovarian Cancer Cells Induced by B-Lactam Steroid Alkylators with Targeted Activity against Poly (ADP-Ribose) Polymerase (PARP) Enzymes in a Cell-Free Assay.
Nikoleousakos N, Dalezis P, Polonifi A, Geromichalou EG, Sagredou S, Alifieris CE, Deligiorgi MV, Sarli V, Trafalis DT.
Nikoleousakos N, et al.
Biomedicines. 2021 Aug 17;9(8):1028. doi: 10.3390/biomedicines9081028.
Biomedicines. 2021.
PMID: 34440232
Free PMC article.
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