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Structure‒tissue exposure/selectivity relationship (STR) correlates with clinical efficacy/safety.
Acta Pharm Sin B. 2022 May;12(5):2462-2478. doi: 10.1016/j.apsb.2022.02.015. Epub 2022 Feb 23.
Acta Pharm Sin B. 2022.
PMID: 35646532
Free PMC article.
Optimization of the Prodrug Moiety of Remdesivir to Improve Lung Exposure/Selectivity and Enhance Anti-SARS-CoV-2 Activity.
Hu H, Mady Traore MD, Li R, Yuan H, He M, Wen B, Gao W, Jonsson CB, Fitzpatrick EA, Sun D.
Hu H, et al. Among authors: mady traore md.
J Med Chem. 2022 Sep 22;65(18):12044-12054. doi: 10.1021/acs.jmedchem.2c00758. Epub 2022 Sep 7.
J Med Chem. 2022.
PMID: 36070561
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A gastrointestinal locally activating Janus kinase inhibitor to treat ulcerative colitis.
Bu Y, Traore MDM, Zhang L, Wang L, Liu Z, Hu H, Wang M, Li C, Sun D.
Bu Y, et al. Among authors: traore mdm.
J Biol Chem. 2023 Dec;299(12):105467. doi: 10.1016/j.jbc.2023.105467. Epub 2023 Nov 17.
J Biol Chem. 2023.
PMID: 37979913
Free PMC article.
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Crossing of the Cystic Barriers of Toxoplasma gondii by the Fluorescent Coumarin Tetra-Cyclopeptide.
Dard C, Leforestier B, Francisco Hilário F, Traoré MDM, Lespinasse MA, Pérès B, Molina MC, Pereira de Freitas R, Milet A, Maubon D, Wong YS.
Dard C, et al. Among authors: traore mdm.
Molecules. 2021 Dec 11;26(24):7506. doi: 10.3390/molecules26247506.
Molecules. 2021.
PMID: 34946588
Free PMC article.
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Synthesis of an Uncharged Tetra-cyclopeptide Acting as a Transmembrane Carrier: Enhanced Cellular and Nuclear Uptake.
Francisco Hilário F, Traoré MD, Zwick V, Berry L, Simões-Pires CA, Cuendet M, Fantozzi N, Pereira de Freitas R, Maynadier M, Wein S, Vial H, Wong YS.
Francisco Hilário F, et al. Among authors: traore md.
Org Lett. 2017 Feb 3;19(3):612-615. doi: 10.1021/acs.orglett.6b03776. Epub 2017 Jan 20.
Org Lett. 2017.
PMID: 28107021
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