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Page 1
Toxicity, pharmacokinetics, and effectiveness of the ortho-chlorinated bispyridinium oxime, K870.
Food Chem Toxicol. 2022 Sep;167:113236. doi: 10.1016/j.fct.2022.113236. Epub 2022 Jun 20.
Food Chem Toxicol. 2022.
PMID: 35738326
A-series agent A-234: initial in vitro and in vivo characterization.
Hrabinova M, Pejchal J, Hepnarova V, Muckova L, Junova L, Opravil J, Zdarova Karasova J, Rozsypal T, Dlabkova A, Rehulkova H, Kucera T, Vecera Z, Caisberger F, Schmidt M, Soukup O, Jun D.
Hrabinova M, et al. Among authors: junova l.
Arch Toxicol. 2024 Apr;98(4):1135-1149. doi: 10.1007/s00204-024-03689-3. Epub 2024 Mar 6.
Arch Toxicol. 2024.
PMID: 38446233
Free PMC article.
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Tacrine - Benzothiazoles: Novel class of potential multitarget anti-Alzheimeŕs drugs dealing with cholinergic, amyloid and mitochondrial systems.
Nepovimova E, Svobodova L, Dolezal R, Hepnarova V, Junova L, Jun D, Korabecny J, Kucera T, Gazova Z, Motykova K, Kubackova J, Bednarikova Z, Janockova J, Jesus C, Cortes L, Pina J, Rostohar D, Serpa C, Soukup O, Aitken L, Hughes RE, Musilek K, Muckova L, Jost P, Chvojkova M, Vales K, Valis M, Chrienova Z, Chalupova K, Kuca K.
Nepovimova E, et al. Among authors: junova l.
Bioorg Chem. 2021 Feb;107:104596. doi: 10.1016/j.bioorg.2020.104596. Epub 2020 Dec 28.
Bioorg Chem. 2021.
PMID: 33421953
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Uncharged mono- and bisoximes: In search of a zwitterion to countermeasure organophosphorus intoxication.
Gorecki L, Markova A, Hepnarova V, Zivna N, Junova L, Hrabinova M, Janousek J, Kobrlova T, Prchal L, Jun D, Soukup O, Horn G, Worek F, Marek J, Korabecny J.
Gorecki L, et al. Among authors: junova l.
Chem Biol Interact. 2024 May 1;394:110941. doi: 10.1016/j.cbi.2024.110941. Epub 2024 Mar 16.
Chem Biol Interact. 2024.
PMID: 38493910
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Tacroximes: novel unique compounds for the recovery of organophosphorus-inhibited acetylcholinesterase.
Gorecki L, Junova L, Kucera T, Hepnarova V, Prchal L, Kobrlova T, Muckova L, Soukup O, Korabecny J.
Gorecki L, et al. Among authors: junova l.
Future Med Chem. 2019 Oct;11(20):2625-2634. doi: 10.4155/fmc-2019-0027. Epub 2019 Sep 26.
Future Med Chem. 2019.
PMID: 31556693
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Synthesis of New Biscoumarin Derivatives, In Vitro Cholinesterase Inhibition, Molecular Modelling and Antiproliferative Effect in A549 Human Lung Carcinoma Cells.
Hudáčová M, Hamuľaková S, Konkoľová E, Jendželovský R, Vargová J, Ševc J, Fedoročko P, Soukup O, Janočková J, Ihnatova V, Kučera T, Bzonek P, Novakova N, Jun D, Junova L, Korábečný J, Kuča K, Kožurková M.
Hudáčová M, et al. Among authors: junova l.
Int J Mol Sci. 2021 Apr 7;22(8):3830. doi: 10.3390/ijms22083830.
Int J Mol Sci. 2021.
PMID: 33917200
Free PMC article.
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Synthesis, Biological Evaluation, and Docking Studies of Novel Bisquaternary Aldoxime Reactivators on Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon.
Kuca K, Jun D, Junova L, Musilek K, Hrabinova M, da Silva JAV, Ramalho TC, Valko M, Wu Q, Nepovimova E, França TCC.
Kuca K, et al. Among authors: junova l.
Molecules. 2018 May 7;23(5):1103. doi: 10.3390/molecules23051103.
Molecules. 2018.
PMID: 29735900
Free PMC article.
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