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kwanghyok son
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Discovery of novel [1,2,4]triazolo[4,3-a]quinoxaline aminophenyl derivatives as BET inhibitors for cancer treatment.
Bioorg Med Chem Lett. 2017 Oct 15;27(20):4606-4613. doi: 10.1016/j.bmcl.2017.09.025. Epub 2017 Sep 14.
Bioorg Med Chem Lett. 2017.
PMID: 28939121
The substantial antiproliferative activities in human cancer cell lines, promising drug-like properties, and the selectivity for the BET family make the lead compound (13) as a novel BRD4 inhibitor motif for anti-cancer drug discovery....
The substantial antiproliferative activities in human cancer cell lines, promising drug-like properties, and the selectivity for the BET …
DW71177: A novel [1,2,4]triazolo[4,3-a]quinoxaline-based potent and BD1-Selective BET inhibitor for the treatment of acute myeloid leukemia.
Ali I, Cha HJ, Lim B, Chae CH, Youm J, Park WJ, Lee SH, Kim JH, Jeong D, Lim JK, Hwang YH, Roe JS, Woo JS, Lee K, Choi G.
Ali I, et al.
Eur J Med Chem. 2024 Feb 5;265:116052. doi: 10.1016/j.ejmech.2023.116052. Epub 2023 Dec 16.
Eur J Med Chem. 2024.
PMID: 38134745
Free article.
The bromodomain and extraterminal domain (BET) family proteins recognize acetyl-lysine (K(ac)) at the histone tail through two tandem bromodomains, i.e., BD1 and BD2, to regulate gene expression. ...
The bromodomain and extraterminal domain (BET) family proteins recognize acetyl-lysine (K(ac)) at the histone tail through two tandem …
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