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2021 | 2 |
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Page 1
Microbial Efflux Pump Inhibitors: A Journey around Quinoline and Indole Derivatives.
Molecules. 2021 Nov 19;26(22):6996. doi: 10.3390/molecules26226996.
Molecules. 2021.
PMID: 34834098
Free PMC article.
Review.
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity.
Nizi MG, Persoons L, Corona A, Felicetti T, Cernicchi G, Massari S, Manfroni G, Vangeel L, Barreca ML, Esposito F, Jochmans D, Milia J, Cecchetti V, Schols D, Neyts J, Tramontano E, Sabatini S, De Jonghe S, Tabarrini O.
Nizi MG, et al. Among authors: cernicchi g.
ACS Med Chem Lett. 2022 May 3;13(5):855-864. doi: 10.1021/acsmedchemlett.2c00123. eCollection 2022 May 12.
ACS Med Chem Lett. 2022.
PMID: 35571875
Free PMC article.
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Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors.
Rampacci E, Felicetti T, Cernicchi G, Stefanetti V, Sabatini S, Passamonti F.
Rampacci E, et al. Among authors: cernicchi g.
Antibiotics (Basel). 2023 Apr 24;12(5):806. doi: 10.3390/antibiotics12050806.
Antibiotics (Basel). 2023.
PMID: 37237709
Free PMC article.
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New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains.
Felicetti T, Cedraro N, Astolfi A, Cernicchi G, Mangiaterra G, Vaiasicca S, Massari S, Manfroni G, Barreca ML, Tabarrini O, Biavasco F, Cecchetti V, Vignaroli C, Sabatini S.
Felicetti T, et al. Among authors: cernicchi g.
Eur J Med Chem. 2022 Nov 5;241:114656. doi: 10.1016/j.ejmech.2022.114656. Epub 2022 Aug 6.
Eur J Med Chem. 2022.
PMID: 35963131
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From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search.
Cedraro N, Cannalire R, Astolfi A, Mangiaterra G, Felicetti T, Vaiasicca S, Cernicchi G, Massari S, Manfroni G, Tabarrini O, Cecchetti V, Barreca ML, Biavasco F, Sabatini S.
Cedraro N, et al. Among authors: cernicchi g.
ChemMedChem. 2021 Oct 6;16(19):3044-3059. doi: 10.1002/cmdc.202100282. Epub 2021 Jun 26.
ChemMedChem. 2021.
PMID: 34032014
Free PMC article.
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