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Year Number of Results
2004 1
2006 1
2008 1
2009 1
2010 1
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2018 3
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Page 1
Novel PD-L1-Targeted Phenyl-Pyrazolone Derivatives with Antioxidant Properties.
Regnault R, Klupsch F, El-Bouazzati H, Magnez R, Le Biannic R, Leleu-Chavain N, Ahouari H, Vezin H, Millet R, Goossens JF, Thuru X, Bailly C. Regnault R, et al. Among authors: klupsch f. Molecules. 2023 Apr 15;28(8):3491. doi: 10.3390/molecules28083491. Molecules. 2023. PMID: 37110727 Free PMC article.
Pyrazolones as inhibitors of immune checkpoint blocking the PD-1/PD-L1 interaction.
Le Biannic R, Magnez R, Klupsch F, Leleu-Chavain N, Thiroux B, Tardy M, El Bouazzati H, Dezitter X, Renault N, Vergoten G, Bailly C, Quesnel B, Thuru X, Millet R. Le Biannic R, et al. Among authors: klupsch f. Eur J Med Chem. 2022 Jun 5;236:114343. doi: 10.1016/j.ejmech.2022.114343. Epub 2022 Apr 4. Eur J Med Chem. 2022. PMID: 35429911
2,6-Diphenylthiazolo[3,2-b][1,2,4]triazoles as telomeric G-quadruplex stabilizers.
El Bakali J, Klupsch F, Guédin A, Brassart B, Fontaine G, Farce A, Roussel P, Houssin R, Bernier JL, Chavatte P, Mergny JL, Riou JF, Hénichart JP. El Bakali J, et al. Among authors: klupsch f. Bioorg Med Chem Lett. 2009 Jul 1;19(13):3434-8. doi: 10.1016/j.bmcl.2009.05.025. Epub 2009 May 12. Bioorg Med Chem Lett. 2009. PMID: 19473838
Synthesis and biological evaluation of ferrocene-based cannabinoid receptor 2 ligands.
Sansook S, Tuo W, Bollier M, Barczyk A, Dezitter X, Klupsch F, Leleu-Chavain N, Farce A, Tizzard GJ, Coles SJ, Spencer J, Millet R. Sansook S, et al. Among authors: klupsch f. Future Med Chem. 2018 Mar 1;10(6):631-638. doi: 10.4155/fmc-2017-0200. Epub 2018 Feb 8. Future Med Chem. 2018. PMID: 29419319 Free article.
One- or Two-Step Synthesis of C-8 and N-9 Substituted Purines.
Bollier M, Klupsch F, Six P, Dubuquoy L, Azaroual N, Millet R, Leleu-Chavain N. Bollier M, et al. Among authors: klupsch f. J Org Chem. 2018 Jan 5;83(1):422-430. doi: 10.1021/acs.joc.7b02269. Epub 2017 Dec 14. J Org Chem. 2018. PMID: 29192784
4-Oxo-1,4-dihydropyridines as selective CB₂ cannabinoid receptor ligands. Part 2: discovery of new agonists endowed with protective effect against experimental colitis.
El Bakali J, Gilleron P, Body-Malapel M, Mansouri R, Muccioli GG, Djouina M, Barczyk A, Klupsch F, Andrzejak V, Lipka E, Furman C, Lambert DM, Chavatte P, Desreumaux P, Millet R. El Bakali J, et al. Among authors: klupsch f. J Med Chem. 2012 Oct 25;55(20):8948-52. doi: 10.1021/jm3008568. Epub 2012 Oct 12. J Med Chem. 2012. PMID: 23017078
13 results