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Page 1
Mental and physical health in family members of substance users: A scoping review.
Drug Alcohol Depend. 2021 Feb 1;219:108439. doi: 10.1016/j.drugalcdep.2020.108439. Epub 2020 Nov 25.
Drug Alcohol Depend. 2021.
PMID: 33333362
Review.
Application of an "inhalation by design" approach to the identification and in-vitro evaluation of novel purine based PI3Kδ inhibitors.
Mazzucato R, Roberti M, Capelli AM, Rancati F, Biagetti M, Fiorelli C, Bruno P, Ronchi P, Bertolini S, Corsi M, Pala D.
Mazzucato R, et al. Among authors: rancati f.
Eur J Med Chem. 2023 Jun 5;254:115331. doi: 10.1016/j.ejmech.2023.115331. Epub 2023 Apr 7.
Eur J Med Chem. 2023.
PMID: 37094451
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Discovery of Clinical Candidate CHF-6366: A Novel Super-soft Dual Pharmacology Muscarinic Antagonist and β2 Agonist (MABA) for the Inhaled Treatment of Respiratory Diseases.
Carzaniga L, Linney ID, Rizzi A, Delcanale M, Schmidt W, Knight CK, Pastore F, Miglietta D, Carnini C, Cesari N, Riccardi B, Mileo V, Venturi L, Moretti E, Blackaby WP, Patacchini R, Accetta A, Biagetti M, Bassani F, Tondelli M, Murgo A, Battipaglia L, Villetti G, Puccini P, Catinella S, Civelli M, Rancati F.
Carzaniga L, et al. Among authors: rancati f.
J Med Chem. 2022 Aug 11;65(15):10233-10250. doi: 10.1021/acs.jmedchem.2c00609. Epub 2022 Jul 28.
J Med Chem. 2022.
PMID: 35901125
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Discovery of a novel class of inhaled dual pharmacology muscarinic antagonist and β2 agonist (MABA) for the treatment of chronic obstructive pulmonary disease (COPD).
Rancati F, Linney ID, Rizzi A, Delcanale M, Knight CK, Schmidt W, Pastore F, Riccardi B, Mileo V, Carnini C, Cesari N, Blackaby WP, Patacchini R, Carzaniga L.
Rancati F, et al.
Bioorg Med Chem Lett. 2021 Jun 1;41:127975. doi: 10.1016/j.bmcl.2021.127975. Epub 2021 Mar 19.
Bioorg Med Chem Lett. 2021.
PMID: 33753262
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Novel Pyrrolidine Derivatives of Budesonide as Long Acting Inhaled Corticosteroids for the Treatment of Pulmonary Inflammatory Diseases.
Ghidini E, Marchini G, Capelli AM, Carnini C, Cenacchi V, Fioni A, Facchinetti F, Rancati F.
Ghidini E, et al. Among authors: rancati f.
J Med Chem. 2018 Jun 14;61(11):4757-4773. doi: 10.1021/acs.jmedchem.7b01873. Epub 2018 May 24.
J Med Chem. 2018.
PMID: 29741897
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Identification of an orally efficacious matrix metalloprotease 12 inhibitor for potential treatment of asthma.
Li W, Li J, Wu Y, Rancati F, Vallese S, Raveglia L, Wu J, Hotchandani R, Fuller N, Cunningham K, Morgan P, Fish S, Krykbaev R, Xu X, Tam S, Goldman SJ, Abraham W, Williams C, Sypek J, Mansour TS.
Li W, et al. Among authors: rancati f.
J Med Chem. 2009 Sep 10;52(17):5408-19. doi: 10.1021/jm900809r.
J Med Chem. 2009.
PMID: 19725580
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Discovery of potent and selective matrix metalloprotease 12 inhibitors for the potential treatment of chronic obstructive pulmonary disease (COPD).
Wu Y, Li J, Wu J, Morgan P, Xu X, Rancati F, Vallese S, Raveglia L, Hotchandani R, Fuller N, Bard J, Cunningham K, Fish S, Krykbaev R, Tam S, Goldman SJ, Williams C, Mansour TS, Saiah E, Sypek J, Li W.
Wu Y, et al. Among authors: rancati f.
Bioorg Med Chem Lett. 2012 Jan 1;22(1):138-43. doi: 10.1016/j.bmcl.2011.11.046. Epub 2011 Nov 20.
Bioorg Med Chem Lett. 2012.
PMID: 22153340
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