Eric R. Samuels - Search Results

Year	Number of Results
2010	1
2013	1
2017	1
2018	3
2019	2
2020	2
2021	2
2022	2
2024	0

1

Allosteric Inhibition of Ubiquitin-like Modifications by a Class of Inhibitor of SUMO-Activating Enzyme.

Li YJ, Du L, Wang J, Vega R, Lee TD, Miao Y, Aldana-Masangkay G, Samuels ER, Li B, Ouyang SX, Colayco SA, Bobkova EV, Divlianska DB, Sergienko E, Chung TDY, Fakih M, Chen Y. Li YJ, et al. Among authors: samuels er. Cell Chem Biol. 2019 Feb 21;26(2):278-288.e6. doi: 10.1016/j.chembiol.2018.10.026. Epub 2018 Dec 20. Cell Chem Biol. 2019. PMID: 30581133 Free PMC article.

2

Photosensitive Ru(II) Complexes as Inhibitors of the Major Human Drug Metabolizing Enzyme CYP3A4.

Toupin N, Steinke SJ, Nadella S, Li A, Rohrabaugh TN Jr, Samuels ER, Turro C, Sevrioukova IF, Kodanko JJ. Toupin N, et al. Among authors: samuels er. J Am Chem Soc. 2021 Jun 23;143(24):9191-9205. doi: 10.1021/jacs.1c04155. Epub 2021 Jun 10. J Am Chem Soc. 2021. PMID: 34110801 Free PMC article.

3

Inhibition of Human CYP3A4 by Rationally Designed Ritonavir-Like Compounds: Impact and Interplay of the Side Group Functionalities.

Samuels ER, Sevrioukova I. Samuels ER, et al. Mol Pharm. 2018 Jan 2;15(1):279-288. doi: 10.1021/acs.molpharmaceut.7b00957. Epub 2017 Dec 12. Mol Pharm. 2018. PMID: 29232137 Free PMC article.

4

Rational Design of CYP3A4 Inhibitors: A One-Atom Linker Elongation in Ritonavir-Like Compounds Leads to a Marked Improvement in the Binding Strength.

Samuels ER, Sevrioukova IF. Samuels ER, et al. Int J Mol Sci. 2021 Jan 16;22(2):852. doi: 10.3390/ijms22020852. Int J Mol Sci. 2021. PMID: 33467005 Free PMC article.

5

An increase in side-group hydrophobicity largely improves the potency of ritonavir-like inhibitors of CYP3A4.

Samuels ER, Sevrioukova IF. Samuels ER, et al. Bioorg Med Chem. 2020 Mar 15;28(6):115349. doi: 10.1016/j.bmc.2020.115349. Epub 2020 Jan 31. Bioorg Med Chem. 2020. PMID: 32044230 Free PMC article.

6

Simultaneous relative UV response determination of known liquid drug product degradants by NMR spectroscopy.

Samuels ER, Wang T. Samuels ER, et al. J Pharm Biomed Anal. 2022 May 10;213:114665. doi: 10.1016/j.jpba.2022.114665. Epub 2022 Feb 17. J Pharm Biomed Anal. 2022. PMID: 35217258

7

Interaction of CYP3A4 with Rationally Designed Ritonavir Analogues: Impact of Steric Constraints Imposed on the Heme-Ligating Group and the End-Pyridine Attachment.

Samuels ER, Sevrioukova IF. Samuels ER, et al. Int J Mol Sci. 2022 Jun 30;23(13):7291. doi: 10.3390/ijms23137291. Int J Mol Sci. 2022. PMID: 35806297 Free PMC article.

8

Direct Synthesis of α-Thio Aromatic Acids from Aromatic Amino Acids.

Samuels ER, Sevrioukova I. Samuels ER, et al. Tetrahedron Lett. 2018 Mar 21;59(12):1140-1142. doi: 10.1016/j.tetlet.2018.02.030. Epub 2018 Feb 13. Tetrahedron Lett. 2018. PMID: 30140110 Free PMC article.

9

Structure-Activity Relationships of Rationally Designed Ritonavir Analogues: Impact of Side-Group Stereochemistry, Headgroup Spacing, and Backbone Composition on the Interaction with CYP3A4.

Samuels ER, Sevrioukova I. Samuels ER, et al. Biochemistry. 2019 Apr 16;58(15):2077-2087. doi: 10.1021/acs.biochem.9b00156. Epub 2019 Apr 3. Biochemistry. 2019. PMID: 30912932 Free PMC article.

10

A microfluidic platform for systems pathology: multiparameter single-cell signaling measurements of clinical brain tumor specimens.

Sun J, Masterman-Smith MD, Graham NA, Jiao J, Mottahedeh J, Laks DR, Ohashi M, DeJesus J, Kamei K, Lee KB, Wang H, Yu ZT, Lu YT, Hou S, Li K, Liu M, Zhang N, Wang S, Angenieux B, Panosyan E, Samuels ER, Park J, Williams D, Konkankit V, Nathanson D, van Dam RM, Phelps ME, Wu H, Liau LM, Mischel PS, Lazareff JA, Kornblum HI, Yong WH, Graeber TG, Tseng HR. Sun J, et al. Among authors: samuels er. Cancer Res. 2010 Aug 1;70(15):6128-38. doi: 10.1158/0008-5472.CAN-10-0076. Epub 2010 Jul 14. Cancer Res. 2010. PMID: 20631065 Free PMC article.

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