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Page 1
Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers.
J Med Chem. 2018 Nov 21;61(22):10155-10172. doi: 10.1021/acs.jmedchem.8b01318. Epub 2018 Oct 31.
J Med Chem. 2018.
PMID: 30339381
Rlf-Mycl Gene Fusion Drives Tumorigenesis and Metastasis in a Mouse Model of Small Cell Lung Cancer.
Ciampricotti M, Karakousi T, Richards AL, Quintanal-Villalonga À, Karatza A, Caeser R, Costa EA, Allaj V, Manoj P, Spainhower KB, Kombak FE, Sanchez-Rivera FJ, Jaspers JE, Zavitsanou AM, Maddalo D, Ventura A, Rideout WM, Akama-Garren EH, Jacks T, Donoghue MTA, Sen T, Oliver TG, Poirier JT, Papagiannakopoulos T, Rudin CM.
Ciampricotti M, et al. Among authors: costa ea.
Cancer Discov. 2021 Dec 1;11(12):3214-3229. doi: 10.1158/2159-8290.CD-21-0441.
Cancer Discov. 2021.
PMID: 34344693
Free PMC article.
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MAPK pathway activation selectively inhibits ASCL1-driven small cell lung cancer.
Caeser R, Hulton C, Costa E, Durani V, Little M, Chen X, Tischfield SE, Asher M, Kombak FE, Chavan SS, Shah NS, Ciampricotti M, de Stanchina E, Poirier JT, Rudin CM, Sen T.
Caeser R, et al. Among authors: costa e.
iScience. 2021 Oct 5;24(11):103224. doi: 10.1016/j.isci.2021.103224. eCollection 2021 Nov 19.
iScience. 2021.
PMID: 34712921
Free PMC article.
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Direct genome editing of patient-derived xenografts using CRISPR-Cas9 enables rapid in vivo functional genomics.
Hulton CH, Costa EA, Shah NS, Quintanal-Villalonga A, Heller G, de Stanchina E, Rudin CM, Poirier JT.
Hulton CH, et al. Among authors: costa ea.
Nat Cancer. 2020 Mar;1(3):359-369. doi: 10.1038/s43018-020-0040-8. Epub 2020 Mar 9.
Nat Cancer. 2020.
PMID: 33345196
Free PMC article.
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Electrochemical advanced oxidation processes as decentralized water treatment technologies to remediate domestic washing machine effluents.
Dos Santos AJ, Costa ECTA, da Silva DR, Garcia-Segura S, Martínez-Huitle CA.
Dos Santos AJ, et al. Among authors: costa ecta.
Environ Sci Pollut Res Int. 2018 Mar;25(7):7002-7011. doi: 10.1007/s11356-017-1039-2. Epub 2017 Dec 22.
Environ Sci Pollut Res Int. 2018.
PMID: 29273989
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