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Page 1
Benzimidazole derivatives endowed with potent antileishmanial activity.
J Enzyme Inhib Med Chem. 2018 Dec;33(1):210-226. doi: 10.1080/14756366.2017.1410480.
J Enzyme Inhib Med Chem. 2018.
PMID: 29233048
Free PMC article.
Quantitative Assessment of Affinity Selection Performance by Using DNA-Encoded Chemical Libraries.
Sannino A, Gabriele E, Bigatti M, Mulatto S, Piazzi J, Scheuermann J, Neri D, Donckele EJ, Samain F.
Sannino A, et al. Among authors: gabriele e.
Chembiochem. 2019 Apr 1;20(7):955-962. doi: 10.1002/cbic.201800766. Epub 2019 Feb 20.
Chembiochem. 2019.
PMID: 30549160
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Optimized Reaction Conditions for Amide Bond Formation in DNA-Encoded Combinatorial Libraries.
Li Y, Gabriele E, Samain F, Favalli N, Sladojevich F, Scheuermann J, Neri D.
Li Y, et al. Among authors: gabriele e.
ACS Comb Sci. 2016 Aug 8;18(8):438-43. doi: 10.1021/acscombsci.6b00058. Epub 2016 Jun 23.
ACS Comb Sci. 2016.
PMID: 27314981
Free PMC article.
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Methanethiosulfonate derivatives as ligands of the STAT3-SH2 domain.
Gabriele E, Ricci C, Meneghetti F, Ferri N, Asai A, Sparatore A.
Gabriele E, et al.
J Enzyme Inhib Med Chem. 2017 Dec;32(1):337-344. doi: 10.1080/14756366.2016.1252757.
J Enzyme Inhib Med Chem. 2017.
PMID: 28097912
Free PMC article.
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Design, Synthesis and In Vitro Investigation of Novel Basic Celastrol Carboxamides as Bio-Inspired Leishmanicidal Agents Endowed with Inhibitory Activity against Leishmania Hsp90.
Bassanini I, Parapini S, Ferrandi EE, Gabriele E, Basilico N, Taramelli D, Sparatore A.
Bassanini I, et al. Among authors: gabriele e.
Biomolecules. 2021 Jan 5;11(1):56. doi: 10.3390/biom11010056.
Biomolecules. 2021.
PMID: 33466300
Free PMC article.
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New sulfurated derivatives of cinnamic acids and rosmaricine as inhibitors of STAT3 and NF-κB transcription factors.
Gabriele E, Brambilla D, Ricci C, Regazzoni L, Taguchi K, Ferri N, Asai A, Sparatore A.
Gabriele E, et al.
J Enzyme Inhib Med Chem. 2017 Dec;32(1):1012-1028. doi: 10.1080/14756366.2017.1350658.
J Enzyme Inhib Med Chem. 2017.
PMID: 28738705
Free PMC article.
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