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Year Number of Results
2012 1
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2019 11
2020 2
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Page 1
Antibacterial activity of noscapine analogs.
Ivanenkov YA, Yu Filyaeva K, Matniyazov RT, Baymiev AK, Baymiev AK, Vladimirova AA, Yamidanov RS, Mavzyutov AR, Zileeva ZR, Zainullina LF, Vakhitova JV, Marina VI, Terentiev VA, Osterman IA, Kartsev VG, Bezrukov DS, Dontsova OA. Ivanenkov YA, et al. Among authors: bezrukov ds. Bioorg Med Chem Lett. 2021 Jul 1;43:128055. doi: 10.1016/j.bmcl.2021.128055. Epub 2021 Apr 21. Bioorg Med Chem Lett. 2021. PMID: 33892103
The Hitchhiker's Guide to Deep Learning Driven Generative Chemistry.
Ivanenkov Y, Zagribelnyy B, Malyshev A, Evteev S, Terentiev V, Kamya P, Bezrukov D, Aliper A, Ren F, Zhavoronkov A. Ivanenkov Y, et al. Among authors: bezrukov d. ACS Med Chem Lett. 2023 Jun 30;14(7):901-915. doi: 10.1021/acsmedchemlett.3c00041. eCollection 2023 Jul 13. ACS Med Chem Lett. 2023. PMID: 37465301 Free PMC article. Review.
2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials.
Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Ayginin AA, Skvortsov DA, Komarova KS, Sadovnikov SV, Matniyazov R, Sofronova AA, Malyshev AS, Machulkin AE, Petrov RA, Lukianov D, Iarovenko S, Bezrukov DS, Baymiev AK, Dontsova OA. Ivanenkov YA, et al. Among authors: bezrukov ds. J Antibiot (Tokyo). 2019 Nov;72(11):827-833. doi: 10.1038/s41429-019-0211-y. Epub 2019 Jul 29. J Antibiot (Tokyo). 2019. PMID: 31358913
Chemistry42: An AI-Driven Platform for Molecular Design and Optimization.
Ivanenkov YA, Polykovskiy D, Bezrukov D, Zagribelnyy B, Aladinskiy V, Kamya P, Aliper A, Ren F, Zhavoronkov A. Ivanenkov YA, et al. Among authors: bezrukov d. J Chem Inf Model. 2023 Feb 13;63(3):695-701. doi: 10.1021/acs.jcim.2c01191. Epub 2023 Feb 2. J Chem Inf Model. 2023. PMID: 36728505 Free PMC article.
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials.
Veselov MS, Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Ayginin AA, Skvortsov DA, Komarova KS, Chemeris AV, Baimiev AK, Sofronova AA, Machulkin AE, Petrov RA, Maklakova SY, Bezrukov DS, Filkov GI, Zainullina LF, Maximova MA, Zileeva ZR, Kartsev VG, Vakhitova YV, Dontsova OA. Veselov MS, et al. Among authors: bezrukov ds. Mol Divers. 2020 Feb;24(1):233-239. doi: 10.1007/s11030-019-09946-3. Epub 2019 Apr 4. Mol Divers. 2020. PMID: 30949901
Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivatives.
Ivanenkov YA, Veselov MS, Rezekin IG, Skvortsov DA, Sandulenko YB, Polyakova MV, Bezrukov DS, Vasilevsky SV, Kukushkin ME, Moiseeva AA, Finko AV, Koteliansky VE, Klyachko NL, Filatova LA, Beloglazkina EK, Zyk NV, Majouga AG. Ivanenkov YA, et al. Among authors: bezrukov ds. Bioorg Med Chem. 2016 Feb 15;24(4):802-11. doi: 10.1016/j.bmc.2015.12.050. Epub 2016 Jan 2. Bioorg Med Chem. 2016. PMID: 26780833
Substituted Furanocoumarins as Novel Class of Antibacterial Translation Inhibitors.
Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Ayginin AA, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Skvortsov DA, Komarova KS, Chemeris AV, Zainullina LF, Maximova MA, Zileeva ZR, Vakhitova YV, Baymiev AK, Baymiev AK, Sofronova AA, Machulkin AE, Petrov RA, Bezrukov DS, Puchinina MM, Lukianov DA, Dontsova OA. Ivanenkov YA, et al. Among authors: bezrukov ds. Comb Chem High Throughput Screen. 2019;22(6):400-410. doi: 10.2174/1386207322666190723110539. Comb Chem High Throughput Screen. 2019. PMID: 31573876
Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA.
Ivanenkov YA, Machulkin AE, Garanina AS, Skvortsov DA, Uspenskaya AA, Deyneka EV, Trofimenko AV, Beloglazkina EK, Zyk NV, Koteliansky VE, Bezrukov DS, Aladinskaya AV, Vorobyeva NS, Puchinina MM, Riabykh GK, Sofronova AA, Malyshev AS, Majouga AG. Ivanenkov YA, et al. Among authors: bezrukov ds. Bioorg Med Chem Lett. 2019 May 15;29(10):1246-1255. doi: 10.1016/j.bmcl.2019.01.040. Epub 2019 Feb 1. Bioorg Med Chem Lett. 2019. PMID: 30904185
Identification of Novel Antibacterials Using Machine Learning Techniques.
Ivanenkov YA, Zhavoronkov A, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Ayginin AA, Kartsev VG, Skvortsov DA, Chemeris AV, Baimiev AK, Sofronova AA, Malyshev AS, Filkov GI, Bezrukov DS, Zagribelnyy BA, Putin EO, Puchinina MM, Dontsova OA. Ivanenkov YA, et al. Among authors: bezrukov ds. Front Pharmacol. 2019 Aug 27;10:913. doi: 10.3389/fphar.2019.00913. eCollection 2019. Front Pharmacol. 2019. PMID: 31507413 Free PMC article.
26 results