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Year Number of Results
2016 2
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2020 5
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2022 3
2023 1
2024 1

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Poly(N-vinylpyrrolidone) Antimalaria Conjugates of Membrane-Disruptive Peptides.
Jokonya S, Langlais M, Leshabane M, Reader PW, Vosloo JA, Pfukwa R, Coertzen D, Birkholtz LM, Rautenbach M, Klumperman B. Jokonya S, et al. Among authors: coertzen d. Biomacromolecules. 2020 Dec 14;21(12):5053-5066. doi: 10.1021/acs.biomac.0c01202. Epub 2020 Nov 6. Biomacromolecules. 2020. PMID: 33156615
The anticancer human mTOR inhibitor sapanisertib potently inhibits multiple Plasmodium kinases and life cycle stages.
Arendse LB, Murithi JM, Qahash T, Pasaje CFA, Godoy LC, Dey S, Gibhard L, Ghidelli-Disse S, Drewes G, Bantscheff M, Lafuente-Monasterio MJ, Fienberg S, Wambua L, Gachuhi S, Coertzen D, van der Watt M, Reader J, Aswat AS, Erlank E, Venter N, Mittal N, Luth MR, Ottilie S, Winzeler EA, Koekemoer LL, Birkholtz LM, Niles JC, Llinás M, Fidock DA, Chibale K. Arendse LB, et al. Among authors: coertzen d. Sci Transl Med. 2022 Oct 19;14(667):eabo7219. doi: 10.1126/scitranslmed.abo7219. Epub 2022 Oct 19. Sci Transl Med. 2022. PMID: 36260689 Free PMC article.
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and In Vivo Efficacy in a Plasmodium berghei Mouse Malaria Infection Model.
Mambwe D, Korkor CM, Mabhula A, Ngqumba Z, Cloete C, Kumar M, Barros PL, Leshabane M, Coertzen D, Taylor D, Gibhard L, Njoroge M, Lawrence N, Reader J, Moreira DR, Birkholtz LM, Wittlin S, Egan TJ, Chibale K. Mambwe D, et al. Among authors: coertzen d. J Med Chem. 2022 Dec 22;65(24):16695-16715. doi: 10.1021/acs.jmedchem.2c01516. Epub 2022 Dec 12. J Med Chem. 2022. PMID: 36507890
Benzimidazole Derivatives Are Potent against Multiple Life Cycle Stages of Plasmodium falciparum Malaria Parasites.
Leshabane M, Dziwornu GA, Coertzen D, Reader J, Moyo P, van der Watt M, Chisanga K, Nsanzubuhoro C, Ferger R, Erlank E, Venter N, Koekemoer L, Chibale K, Birkholtz LM. Leshabane M, et al. Among authors: coertzen d. ACS Infect Dis. 2021 Jul 9;7(7):1945-1955. doi: 10.1021/acsinfecdis.0c00910. Epub 2021 Mar 5. ACS Infect Dis. 2021. PMID: 33673735 Free article.
Antimalarial Benzimidazole Derivatives Incorporating Phenolic Mannich Base Side Chains Inhibit Microtubule and Hemozoin Formation: Structure-Activity Relationship and In Vivo Oral Efficacy Studies.
Dziwornu GA, Coertzen D, Leshabane M, Korkor CM, Cloete CK, Njoroge M, Gibhard L, Lawrence N, Reader J, van der Watt M, Wittlin S, Birkholtz LM, Chibale K. Dziwornu GA, et al. Among authors: coertzen d. J Med Chem. 2021 Apr 22;64(8):5198-5215. doi: 10.1021/acs.jmedchem.1c00354. Epub 2021 Apr 12. J Med Chem. 2021. PMID: 33844521
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of Plasmodium Phosphatidylinositol-4-kinase and cGMP-Dependent Protein Kinase.
Cheuka PM, Centani L, Arendse LB, Fienberg S, Wambua L, Renga SS, Dziwornu GA, Kumar M, Lawrence N, Taylor D, Wittlin S, Coertzen D, Reader J, van der Watt M, Birkholtz LM, Chibale K. Cheuka PM, et al. Among authors: coertzen d. ACS Infect Dis. 2021 Jan 8;7(1):34-46. doi: 10.1021/acsinfecdis.0c00481. Epub 2020 Dec 15. ACS Infect Dis. 2021. PMID: 33319990
21 results