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2018 2
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The 1,8-naphthyridines sulfonamides are NorA efflux pump inhibitors.
Oliveira-Tintino CDM, Muniz DF, Barbosa CRDS, Pereira RLS, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Pereira PS, Costa JGMD, Rodrigues FFG, Teixeira AMR, Ribeiro-Filho J, Tintino SR, de Menezes IRA, Coutinho HDM, Silva TGD. Oliveira-Tintino CDM, et al. J Glob Antimicrob Resist. 2021 Mar;24:233-240. doi: 10.1016/j.jgar.2020.11.027. Epub 2020 Dec 29. J Glob Antimicrob Resist. 2021. PMID: 33385589 Free article.
Liposome evaluation in inhibiting pump efflux of NorA of Staphylococcus aureus.
Júnior JGAS, Coutinho HDM, Rodrigues JPV, Ferreira VPG, Neto JBA, Costa da Silva MM, Justino de Araújo AC, Pereira RLS, Alexandre de Aquino PE, Oliveira-Tintino CDM, Nicolete R. Júnior JGAS, et al. Chem Phys Lipids. 2022 Jul;245:105204. doi: 10.1016/j.chemphyslip.2022.105204. Epub 2022 Apr 7. Chem Phys Lipids. 2022. PMID: 35398337
3-Substituted Coumarins Inhibit NorA and MepA Efflux Pumps of Staphylococcus aureus.
Araújo-Neto JB, Oliveira-Tintino CDM, de Araújo GA, Alves DS, Ribeiro FR, Brancaglion GA, Carvalho DT, Lima CMG, Mohammed Ali HSH, Rather IA, Wani MY, Emran TB, Coutinho HDM, Balbino VQ, Tintino SR. Araújo-Neto JB, et al. Among authors: oliveira tintino cdm. Antibiotics (Basel). 2023 Dec 15;12(12):1739. doi: 10.3390/antibiotics12121739. Antibiotics (Basel). 2023. PMID: 38136773 Free PMC article.
Enhancement of Antibiotic Activity by 1,8-Naphthyridine Derivatives against Multi-Resistant Bacterial Strains.
Araújo-Neto JB, Silva MMCD, Oliveira-Tintino CDM, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Ribeiro-Filho J, Siyadatpanah A, Wilairatana P, Coutinho HDM, Tintino SR. Araújo-Neto JB, et al. Among authors: oliveira tintino cdm. Molecules. 2021 Dec 6;26(23):7400. doi: 10.3390/molecules26237400. Molecules. 2021. PMID: 34885981 Free PMC article.
In vitro evaluation of the susceptibility of bacterial biofilms to hecogenin acetate.
Araújo NJS, Costa MDS, da Silva ARP, Paulo CLR, Silva CAP, Felix FJ, Oliveira-Tintino CDM, Filho JMB, de Freitas TS, Braga MFBM, Coutinho HDM, Andrade-Pinheiro JC. Araújo NJS, et al. Acta Trop. 2024 May;253:107157. doi: 10.1016/j.actatropica.2024.107157. Epub 2024 Feb 22. Acta Trop. 2024. PMID: 38387772
Modification of Antibiotic Activity by Fixed Oil of the Artocarpus heterophyllus Almond against Standard and Multidrug-Resistant Bacteria Strains.
Dias CJF, Raposo A, de Sousa CDT, de Araújo-Neto JB, Tintino SR, Oliveira-Tintino CDM, Araújo IM, Coutinho HDM, Costa MGM, Lima CG, de Alencar MS, Carrascosa C, Saraiva A, de Sousa EO. Dias CJF, et al. Biology (Basel). 2022 Dec 16;11(12):1835. doi: 10.3390/biology11121835. Biology (Basel). 2022. PMID: 36552343 Free PMC article.
Chemical synthesis, molecular docking and MepA efflux pump inhibitory effect by 1,8-naphthyridines sulfonamides.
Oliveira-Tintino CDM, Tintino SR, Muniz DF, Rodrigues Dos Santos Barbosa C, Pereira RLS, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Krautler MIL, Pereira PS, Balbino TCL, da Costa JGM, Rodrigues FFG, Teixeira AMR, Barreto HM, de Menezes IRA, Coutinho HDM, da Silva TG. Oliveira-Tintino CDM, et al. Eur J Pharm Sci. 2021 May 1;160:105753. doi: 10.1016/j.ejps.2021.105753. Epub 2021 Feb 10. Eur J Pharm Sci. 2021. PMID: 33581258
Efflux Pump (QacA, QacB, and QacC) and β-Lactamase Inhibitors? An Evaluation of 1,8-Naphthyridines against Staphylococcus aureus Strains.
Oliveira-Tintino CDM, Tintino SR, Justino de Araújo AC, Dos Santos Barbosa CR, Ramos Freitas P, Araújo Neto JB, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Barreto HM, Ribeiro-Filho J, de Menezes IRA, Coutinho HDM. Oliveira-Tintino CDM, et al. Molecules. 2023 Feb 15;28(4):1819. doi: 10.3390/molecules28041819. Molecules. 2023. PMID: 36838807 Free PMC article.
22 results