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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
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2016 | 1 |
2018 | 2 |
2020 | 1 |
2021 | 1 |
2022 | 1 |
2024 | 0 |
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Page 1
Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria.
Pharmaceuticals (Basel). 2022 Jun 20;15(6):766. doi: 10.3390/ph15060766.
Pharmaceuticals (Basel). 2022.
PMID: 35745685
Free PMC article.
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor.
Magalhães J, Franko N, Raboni S, Annunziato G, Tammela P, Bruno A, Bettati S, Mozzarelli A, Pieroni M, Campanini B, Costantino G.
Magalhães J, et al. Among authors: bruno a.
ACS Med Chem Lett. 2020 Feb 13;11(5):790-797. doi: 10.1021/acsmedchemlett.9b00627. eCollection 2020 May 14.
ACS Med Chem Lett. 2020.
PMID: 32435386
Free PMC article.
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Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants.
Magalhães J, Franko N, Raboni S, Annunziato G, Tammela P, Bruno A, Bettati S, Armao S, Spadini C, Cabassi CS, Mozzarelli A, Pieroni M, Campanini B, Costantino G.
Magalhães J, et al. Among authors: bruno a.
Pharmaceuticals (Basel). 2021 Feb 23;14(2):174. doi: 10.3390/ph14020174.
Pharmaceuticals (Basel). 2021.
PMID: 33672408
Free PMC article.
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Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets.
Magalhães J, Annunziato G, Franko N, Pieroni M, Campanini B, Bruno A, Costantino G.
Magalhães J, et al. Among authors: bruno a.
J Chem Inf Model. 2018 Mar 26;58(3):710-723. doi: 10.1021/acs.jcim.7b00733. Epub 2018 Mar 6.
J Chem Inf Model. 2018.
PMID: 29481752
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Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug design.
Magalhães J, Franko N, Annunziato G, Welch M, Dolan SK, Bruno A, Mozzarelli A, Armao S, Jirgensons A, Pieroni M, Costantino G, Campanini B.
Magalhães J, et al. Among authors: bruno a.
J Enzyme Inhib Med Chem. 2018 Dec;33(1):1444-1452. doi: 10.1080/14756366.2018.1512596.
J Enzyme Inhib Med Chem. 2018.
PMID: 30221554
Free PMC article.
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Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR.
Annunziato G, Pieroni M, Benoni R, Campanini B, Pertinhez TA, Pecchini C, Bruno A, Magalhães J, Bettati S, Franko N, Mozzarelli A, Costantino G.
Annunziato G, et al. Among authors: bruno a.
J Enzyme Inhib Med Chem. 2016;31(sup4):78-87. doi: 10.1080/14756366.2016.1218486. Epub 2016 Aug 31.
J Enzyme Inhib Med Chem. 2016.
PMID: 27578398
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