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2021 | 2 |
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Page 1
Synthetic Heterocyclic Derivatives as Kinase Inhibitors Tested for the Treatment of Neuroblastoma.
Molecules. 2021 Nov 23;26(23):7069. doi: 10.3390/molecules26237069.
Molecules. 2021.
PMID: 34885651
Free PMC article.
Review.
Identification and Biological Characterization of the Pyrazolo[3,4-d]pyrimidine Derivative SI388 Active as Src Inhibitor.
Contadini C, Cirotti C, Carbone A, Norouzi M, Cianciusi A, Crespan E, Perini C, Maga G, Barilà D, Musumeci F, Schenone S.
Contadini C, et al. Among authors: cianciusi a.
Pharmaceuticals (Basel). 2023 Jul 4;16(7):958. doi: 10.3390/ph16070958.
Pharmaceuticals (Basel). 2023.
PMID: 37513870
Free PMC article.
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Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment.
Di Maria S, Picarazzi F, Mori M, Cianciusi A, Carbone A, Crespan E, Perini C, Sabetta S, Deplano S, Poggialini F, Molinari A, Aronne R, Maccioni E, Maga G, Angelucci A, Schenone S, Musumeci F, Dreassi E.
Di Maria S, et al. Among authors: cianciusi a.
Bioorg Chem. 2022 Nov;128:106071. doi: 10.1016/j.bioorg.2022.106071. Epub 2022 Aug 1.
Bioorg Chem. 2022.
PMID: 35932498
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Si113-prodrugs selectively activated by plasmin against hepatocellular and ovarian carcinoma.
Rango E, D'Antona L, Iovenitti G, Brai A, Mancini A, Zamperini C, Trivisani CI, Marianelli S, Fallacara AL, Molinari A, Cianciusi A, Schenone S, Perrotti N, Dreassi E, Botta M.
Rango E, et al. Among authors: cianciusi a.
Eur J Med Chem. 2021 Nov 5;223:113653. doi: 10.1016/j.ejmech.2021.113653. Epub 2021 Jun 17.
Eur J Med Chem. 2021.
PMID: 34161866
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Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment.
Vagaggini C, Petroni D, D'Agostino I, Poggialini F, Cavallini C, Cianciusi A, Salis A, D'Antona L, Francesconi V, Manetti F, Damonte G, Musumeci F, Menichetti L, Dreassi E, Carbone A, Schenone S.
Vagaggini C, et al. Among authors: cianciusi a.
Drug Dev Res. 2024 Feb;85(1):e22158. doi: 10.1002/ddr.22158.
Drug Dev Res. 2024.
PMID: 38349262
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