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Year Number of Results
2019 1
2020 7
2021 13
2022 11
2023 5
2024 3

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Page 1
Potentiating activity of Norfloxacin by synthetic chalcones against NorA overproducing Staphylococcus aureus.
Alves Borges Leal AL, Teixeira da Silva P, Nunes da Rocha M, Marinho EM, Marinho ES, Marinho MM, Bandeira PN, Sampaio Nogueira CE, Barreto HM, Rodrigues Teixeira AM, Silva Dos Santos H. Alves Borges Leal AL, et al. Among authors: rodrigues teixeira am. Microb Pathog. 2021 Jun;155:104894. doi: 10.1016/j.micpath.2021.104894. Epub 2021 Apr 21. Microb Pathog. 2021. PMID: 33894291 Review.
NorA, Tet(K), MepA, and MsrA Efflux Pumps in Staphylococcus aureus, their Inhibitors and 1,8-Naphthyridine Sulfonamides.
de Morais Oliveira-Tintino CD, Muniz DF, Dos Santos Barbosa CR, Silva Pereira RL, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Lacowicz Krautler MI, Barros Oliveira CV, Pereira PS, Rodrigues Teixeira AM, Tintino SR, de Menezes IRA, Melo Coutinho HD, da Silva TG. de Morais Oliveira-Tintino CD, et al. Among authors: rodrigues teixeira am. Curr Pharm Des. 2023;29(5):323-355. doi: 10.2174/1381612829666221212101501. Curr Pharm Des. 2023. PMID: 36515045 Review.
Potentiation of antibiotic activity, and efflux pumps inhibition by (2E)-1-(4-aminophenyl)-3-(4-fluorophenyl)prop-2-en-1-one.
Hemília de Souza Nunes P, Sampaio de Freitas T, Esmeraldo Rocha J, Luiz Silva Pereira R, Machado Marinho M, de Oliveira MR, Santos Oliveira L, Machado Marinho E, Silva Marinho E, Sousa Aquino S, Emidio Sampaio Nogueira C, Douglas Melo Coutinho H, Nogueira Bandeira P, Magno Rodrigues Teixeira A, Dos Santos HS. Hemília de Souza Nunes P, et al. Among authors: magno rodrigues teixeira a. Fundam Clin Pharmacol. 2022 Dec;36(6):1066-1082. doi: 10.1111/fcp.12785. Epub 2022 May 19. Fundam Clin Pharmacol. 2022. PMID: 35475507
The 1,8-naphthyridines sulfonamides are NorA efflux pump inhibitors.
Oliveira-Tintino CDM, Muniz DF, Barbosa CRDS, Pereira RLS, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Pereira PS, Costa JGMD, Rodrigues FFG, Teixeira AMR, Ribeiro-Filho J, Tintino SR, de Menezes IRA, Coutinho HDM, Silva TGD. Oliveira-Tintino CDM, et al. Among authors: teixeira amr. J Glob Antimicrob Resist. 2021 Mar;24:233-240. doi: 10.1016/j.jgar.2020.11.027. Epub 2020 Dec 29. J Glob Antimicrob Resist. 2021. PMID: 33385589 Free article.
GABAA receptor participation in anxiolytic and anticonvulsant effects of (E)-3-(furan-2-yl)-1-(2hydroxy-3,4,6-trimethoxyphenyl)prop-2-en-1-one in adult zebrafish.
Silva Mendes FR, Wlisses da Silva A, Amâncio Ferreira MK, de Lima Rebouças E, Marinho EM, Marinho MM, Bandeira PN, Rodrigues Teixeira AM, Silva Alencar de Menezes JE, Alves de Siqueira E, Róseo Paula Pessoa Bezerra de Menezes R, Marinho ES, Silva Dos Santos H. Silva Mendes FR, et al. Among authors: rodrigues teixeira am. Neurochem Int. 2022 May;155:105303. doi: 10.1016/j.neuint.2022.105303. Epub 2022 Feb 17. Neurochem Int. 2022. PMID: 35183661
Aminophenyl chalcones potentiating antibiotic activity and inhibiting bacterial efflux pump.
Siqueira MMR, Freire PTC, Cruz BG, de Freitas TS, Bandeira PN, Silva Dos Santos H, Nogueira CES, Teixeira AMR, Pereira RLS, Xavier JDC, Campina FF, Dos Santos Barbosa CR, Neto JBA, da Silva MMC, Siqueira-Júnior JP, Douglas Melo Coutinho H. Siqueira MMR, et al. Among authors: teixeira amr. Eur J Pharm Sci. 2021 Mar 1;158:105695. doi: 10.1016/j.ejps.2020.105695. Epub 2020 Dec 29. Eur J Pharm Sci. 2021. PMID: 33383131
Chloride substitution on 2-hydroxy-3,4,6-trimethoxyphenylchalcones improves in vitro selectivity on Trypanosoma cruzi strain Y.
Magalhães EP, Gomes NDB, Freitas TA, Silva BP, Ribeiro LR, Ameida-Neto FWQ, Marinho MM, Lima-Neto P, Marinho ES, Santos HSD, Teixeira AMR, Sampaio TL, Menezes RRPPB, Martins AMC. Magalhães EP, et al. Among authors: teixeira amr. Chem Biol Interact. 2022 Jul 1;361:109920. doi: 10.1016/j.cbi.2022.109920. Epub 2022 Apr 21. Chem Biol Interact. 2022. PMID: 35461787
In silico study of the potential interactions of 4'-acetamidechalcones with protein targets in SARS-CoV-2.
Q Almeida-Neto FW, Castro Matos MG, Marinho EM, Marinho MM, Róseo Paula Pessoa Bezerra de Menezes R, Sampaio TL, Bandeira PN, Celedonio Fernandes CF, Magno Rodrigues Teixeira A, Marinho ES, de Lima-Neto P, Silva Dos Santos H. Q Almeida-Neto FW, et al. Among authors: magno rodrigues teixeira a. Biochem Biophys Res Commun. 2021 Jan 22;537:71-77. doi: 10.1016/j.bbrc.2020.12.074. Epub 2020 Dec 26. Biochem Biophys Res Commun. 2021. PMID: 33387885 Free PMC article.
Chemical synthesis, molecular docking and MepA efflux pump inhibitory effect by 1,8-naphthyridines sulfonamides.
Oliveira-Tintino CDM, Tintino SR, Muniz DF, Rodrigues Dos Santos Barbosa C, Pereira RLS, Begnini IM, Rebelo RA, da Silva LE, Mireski SL, Nasato MC, Krautler MIL, Pereira PS, Balbino TCL, da Costa JGM, Rodrigues FFG, Teixeira AMR, Barreto HM, de Menezes IRA, Coutinho HDM, da Silva TG. Oliveira-Tintino CDM, et al. Among authors: teixeira amr. Eur J Pharm Sci. 2021 May 1;160:105753. doi: 10.1016/j.ejps.2021.105753. Epub 2021 Feb 10. Eur J Pharm Sci. 2021. PMID: 33581258
31 results