Desrayaud S - Search Results

1

Developing Low Molecular Weight PET and SPECT Imaging Agents.

Xue L, Jie CVML, Desrayaud S, Auberson YP. Xue L, et al. Among authors: desrayaud s. ChemMedChem. 2024 Apr 18:e202400094. doi: 10.1002/cmdc.202400094. Online ahead of print. ChemMedChem. 2024. PMID: 38634545 Review.

2

Improving In Vitro-In Vivo Extrapolation of Clearance Using Rat Liver Microsomes for Highly Plasma Protein-Bound Molecules.

Trunzer M, Teigão J, Huth F, Poller B, Desrayaud S, Rodríguez-Pérez R, Faller B. Trunzer M, et al. Among authors: desrayaud s. Drug Metab Dispos. 2024 Apr 16;52(5):345-354. doi: 10.1124/dmd.123.001597. Drug Metab Dispos. 2024. PMID: 38360916

3

Discovery of Potent, Orally Bioavailable, Tricyclic NLRP3 Inhibitors.

Velcicky J, Janser P, Gommermann N, Brenneisen S, Ilic S, Vangrevelinghe E, Stiefl N, Boettcher A, Arnold C, Malinverni C, Dawson J, Murgasova R, Desrayaud S, Beltz K, Hinniger A, Dekker C, Farady CJ, Mackay A. Velcicky J, et al. Among authors: desrayaud s. J Med Chem. 2024 Jan 25;67(2):1544-1562. doi: 10.1021/acs.jmedchem.3c02098. Epub 2024 Jan 4. J Med Chem. 2024. PMID: 38175811

4

A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system.

Auberson YP, Lièvre A, Desrayaud S, Briard E. Auberson YP, et al. Among authors: desrayaud s. J Labelled Comp Radiopharm. 2022 Nov;65(13):343-350. doi: 10.1002/jlcr.4004. Epub 2022 Sep 29. J Labelled Comp Radiopharm. 2022. PMID: 36148533

5

Predicting In Vivo Compound Brain Penetration Using Multi-task Graph Neural Networks.

Hamzic S, Lewis R, Desrayaud S, Soylu C, Fortunato M, Gerebtzoff G, Rodríguez-Pérez R. Hamzic S, et al. Among authors: desrayaud s. J Chem Inf Model. 2022 Jul 11;62(13):3180-3190. doi: 10.1021/acs.jcim.2c00412. Epub 2022 Jun 23. J Chem Inf Model. 2022. PMID: 35738004 Review.

6

Identification of NVP-CLR457 as an Orally Bioavailable Non-CNS-Penetrant pan-Class IA Phosphoinositol-3-Kinase Inhibitor.

Fairhurst RA, Furet P, Imbach-Weese P, Stauffer F, Rueeger H, McCarthy C, Ripoche S, Oswald S, Arnaud B, Jary A, Maira M, Schnell C, Guthy DA, Wartmann M, Kiffe M, Desrayaud S, Blasco F, Widmer T, Seiler F, Gutmann S, Knapp M, Caravatti G. Fairhurst RA, et al. Among authors: desrayaud s. J Med Chem. 2022 Jun 23;65(12):8345-8379. doi: 10.1021/acs.jmedchem.2c00267. Epub 2022 May 2. J Med Chem. 2022. PMID: 35500094

7

Modulation of Oral Bioavailability and Metabolism for Closely Related Cyclic Hexapeptides.

Vorherr T, Lewis I, Berghausen J, Desrayaud S, Schaefer M. Vorherr T, et al. Among authors: desrayaud s. Int J Pept Res Ther. 2018;24(1):35-48. doi: 10.1007/s10989-017-9590-8. Epub 2017 Mar 28. Int J Pept Res Ther. 2018. PMID: 29527142 Free PMC article.

8

Brain region-specific enhancement of remyelination and prevention of demyelination by the CSF1R kinase inhibitor BLZ945.

Beckmann N, Giorgetti E, Neuhaus A, Zurbruegg S, Accart N, Smith P, Perdoux J, Perrot L, Nash M, Desrayaud S, Wipfli P, Frieauff W, Shimshek DR. Beckmann N, et al. Among authors: desrayaud s. Acta Neuropathol Commun. 2018 Feb 15;6(1):9. doi: 10.1186/s40478-018-0510-8. Acta Neuropathol Commun. 2018. PMID: 29448957 Free PMC article.

9

Utility of food pellets containing 1-aminobenzotriazole for longer term in vivo inhibition of cytochrome P450 in mice.

Stringer R, Cordier V, Afatsawo C, Arabin P, Desrayaud S, Hoffmann L, Lehmann D, Lowe PJ, Risser F, Thiel J, Widmer T, Wipfli P, Bigaud M. Stringer R, et al. Among authors: desrayaud s. Xenobiotica. 2019 Jan;49(1):13-21. doi: 10.1080/00498254.2017.1418542. Epub 2018 Jan 29. Xenobiotica. 2019. PMID: 29299977

10

Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist.

Orain D, Tasdelen E, Haessig S, Koller M, Picard A, Dubois C, Lingenhoehl K, Desrayaud S, Floersheim P, Carcache D, Urwyler S, Kallen J, Mattes H. Orain D, et al. Among authors: desrayaud s. ChemMedChem. 2017 Feb 3;12(3):197-201. doi: 10.1002/cmdc.201600467. Epub 2016 Nov 15. ChemMedChem. 2017. PMID: 27863026

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