Wróbel TM - Search Results

1

Discovery and in vitro Evaluation of Novel Serotonin 5-HT2A Receptor Ligands Identified Through Virtual Screening.

Zięba A, Bartuzi D, Stępnicki P, Matosiuk D, Wróbel TM, Laitinen T, Castro M, Kaczor AA. Zięba A, et al. Among authors: wrobel tm. ChemMedChem. 2024 Apr 15:e202400080. doi: 10.1002/cmdc.202400080. Online ahead of print. ChemMedChem. 2024. PMID: 38619283

2

Synthesis and molecular docking of novel non-competitive antagonists of GluK2 receptor.

Kaczor AA, Wróbel T, Kronbach C, Unverferth K, Stachal T, Matosiuk D. Kaczor AA, et al. Med Chem Res. 2015;24(2):810-817. doi: 10.1007/s00044-014-1171-1. Epub 2014 Jul 24. Med Chem Res. 2015. PMID: 25620864 Free PMC article.

3

Synthesis, pharmacological and structural studies of 5-substituted-3-(1-arylmethyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indoles as multi-target ligands of aminergic GPCRs.

Kondej M, Wróbel TM, Silva AG, Stępnicki P, Koszła O, Kędzierska E, Bartyzel A, Biała G, Matosiuk D, Loza MI, Castro M, Kaczor AA. Kondej M, et al. Among authors: wrobel tm. Eur J Med Chem. 2019 Oct 15;180:673-689. doi: 10.1016/j.ejmech.2019.07.050. Epub 2019 Jul 20. Eur J Med Chem. 2019. PMID: 31357129

4

Tuning Down the Pain - An Overview of Allosteric Modulation of Opioid Receptors: Mechanisms of Modulation, Allosteric Sites, Modulator Syntheses.

Bartuzi D, Wróbel TM, Kaczor AA, Matosiuk D. Bartuzi D, et al. Among authors: wrobel tm. Curr Top Med Chem. 2020;20(31):2852-2865. doi: 10.2174/1568026620666200601155451. Curr Top Med Chem. 2020. PMID: 32479245 Review.

5

Allosteric modulation of dopamine D_2L receptor in complex with G_i1 and G_i2 proteins: the effect of subtle structural and stereochemical ligand modifications.

Żuk J, Bartuzi D, Silva AG, Pitucha M, Koszła O, Wróbel TM, Matosiuk D, Castro M, Kaczor AA. Żuk J, et al. Among authors: wrobel tm. Pharmacol Rep. 2022 Apr;74(2):406-424. doi: 10.1007/s43440-021-00352-x. Epub 2022 Jan 22. Pharmacol Rep. 2022. PMID: 35064921 Free PMC article.

6

WaterMap-Guided Structure-Based Virtual Screening for Acetylcholinesterase Inhibitors.

Targowska-Duda KM, Maj M, Drączkowski P, Budzyńska B, Boguszewska-Czubara A, Wróbel TM, Laitinen T, Kaczmar P, Poso A, Kaczor AA. Targowska-Duda KM, et al. Among authors: wrobel tm. ChemMedChem. 2022 Apr 20;17(8):e202100721. doi: 10.1002/cmdc.202100721. Epub 2022 Mar 4. ChemMedChem. 2022. PMID: 35157366

7

Multitarget Derivatives of D2AAK1 as Potential Antipsychotics: The Effect of Substitution in the Indole Moiety.

Kondej M, Wróbel TM, Targowska-Duda KM, Leandro Martínez A, Koszła O, Stępnicki P, Zięba A, Paz A, Wronikowska-Denysiuk O, Loza MI, Castro M, Kaczor AA. Kondej M, et al. Among authors: wrobel tm. ChemMedChem. 2022 Aug 3;17(15):e202200238. doi: 10.1002/cmdc.202200238. Epub 2022 Jun 17. ChemMedChem. 2022. PMID: 35610178

8

Funnel metadynamics and behavioral studies reveal complex effect of D2AAK1 ligand on anxiety-like processes.

Bartuzi D, Kędzierska E, Targowska-Duda KM, Koszła O, Wróbel TM, Jademyr S, Karcz T, Szczepańska K, Stępnicki P, Wronikowska-Denysiuk O, Biała G, Handzlik J, Kristensen JL, Poso A, Kaczor AA. Bartuzi D, et al. Among authors: wrobel tm. Sci Rep. 2022 Dec 7;12(1):21192. doi: 10.1038/s41598-022-25478-7. Sci Rep. 2022. PMID: 36476619 Free PMC article.

9

Allosteric Modulators of Dopamine D₂ Receptors for Fine-Tuning of Dopaminergic Neurotransmission in CNS Diseases: Overview, Pharmacology, Structural Aspects and Synthesis.

Kaczor AA, Wróbel TM, Bartuzi D. Kaczor AA, et al. Among authors: wrobel tm. Molecules. 2022 Dec 25;28(1):178. doi: 10.3390/molecules28010178. Molecules. 2022. PMID: 36615372 Free PMC article. Review.

10

Synthesis, Structural and Behavioral Studies of Indole Derivatives D2AAK5, D2AAK6 and D2AAK7 as Serotonin 5-HT_1A and 5-HT_2A Receptor Ligands.

Kaczor AA, Kędzierska E, Wróbel TM, Grudzińska A, Pawlak A, Laitinen T, Bartyzel A. Kaczor AA, et al. Among authors: wrobel tm. Molecules. 2023 Jan 2;28(1):383. doi: 10.3390/molecules28010383. Molecules. 2023. PMID: 36615578 Free PMC article.

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