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First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer's Disease.
Santini A, Tassinari E, Poeta E, Loi M, Ciani E, Trazzi S, Piccarducci R, Daniele S, Martini C, Pagliarani B, Tarozzi A, Bersani M, Spyrakis F, Danková D, Olsen CA, Soldati R, Tumiatti V, Montanari S, De Simone A, Milelli A. Santini A, et al. Among authors: piccarducci r. ACS Chem Neurosci. 2024 May 15. doi: 10.1021/acschemneuro.4c00061. Online ahead of print. ACS Chem Neurosci. 2024. PMID: 38747979
Development and Nanoparticle-Mediated Delivery of Novel MDM2/MDM4 Heterodimer Peptide Inhibitors to Enhance 5-Fluorouracil Nucleolar Stress in Colorectal Cancer Cells.
Merlino F, Pecoraro A, Longobardi G, Donati G, Di Leva FS, Brignola C, Piccarducci R, Daniele S, Martini C, Marinelli L, Russo G, Quaglia F, Conte C, Russo A, La Pietra V. Merlino F, et al. Among authors: piccarducci r. J Med Chem. 2024 Feb 8;67(3):1812-1824. doi: 10.1021/acs.jmedchem.3c01312. Epub 2024 Jan 29. J Med Chem. 2024. PMID: 38285632
Apolipoprotein E ε4 triggers neurotoxicity via cholesterol accumulation, acetylcholine dyshomeostasis, and PKCε mislocalization in cholinergic neuronal cells.
Piccarducci R, Giacomelli C, Bertilacchi MS, Benito-Martinez A, Di Giorgi N, Daniele S, Signore G, Rocchiccioli S, Vilar M, Marchetti L, Martini C. Piccarducci R, et al. Biochim Biophys Acta Mol Basis Dis. 2023 Oct;1869(7):166793. doi: 10.1016/j.bbadis.2023.166793. Epub 2023 Jun 17. Biochim Biophys Acta Mol Basis Dis. 2023. PMID: 37336366 Free article.
Intermittent hypoxia treatments cause cellular priming in human microglia.
De Felice M, Germelli L, Piccarducci R, Da Pozzo E, Giacomelli C, Baccaglini-Frank A, Martini C. De Felice M, et al. Among authors: piccarducci r. J Cell Mol Med. 2023 Mar;27(6):819-830. doi: 10.1111/jcmm.17682. Epub 2023 Feb 23. J Cell Mol Med. 2023. PMID: 36824025 Free PMC article.
α-synuclein as an emerging pathophysiological biomarker of Alzheimer's disease.
Beatino MF, De Luca C, Campese N, Belli E, Piccarducci R, Giampietri L, Martini C, Perugi G, Siciliano G, Ceravolo R, Vergallo A, Hampel H, Baldacci F. Beatino MF, et al. Among authors: piccarducci r. Expert Rev Mol Diagn. 2022 Apr;22(4):411-425. doi: 10.1080/14737159.2022.2068952. Epub 2022 May 6. Expert Rev Mol Diagn. 2022. PMID: 35443850 Review.
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